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2-(3-{1-[(6-methylpyridin-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-4-(trifluoromethyl)pyrimidine
(2R,6R)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[(1-acetylpiperidin-4-yl)methyl]-5-(thiophen-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-(2-aminoethyl)-4-(naphthalen-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,8aR)-6-(6-aminopyrimidin-4-yl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-({cyclopropyl[(2-ethoxyphenyl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{4-[2-(azepane-1-carbonyl)-4-chlorophenoxy]piperidin-1-yl}ethan-1-one
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrrolidin-2-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-[3-(4-{[2-(1H-imidazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
N-methyl-5-(5-propyl-1,2-oxazole-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
2-(propan-2-yl)-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-2,5-dihydro-1H-pyrrole
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
1-ethyl-4-{[methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amino]methyl}pyrrolidin-2-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-acetamido-3-methylbutanamide
(2R,6S)-2,6-dimethyl-4-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)morpholine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[ethyl({[(3S,4R)-4-(hydroxymethyl)-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
4-(hydroxymethyl)-1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-4-ol
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(4-methoxyphenoxymethyl)piperidine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}benzamide
(2S)-2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidine
4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)butanamide
N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
1-(2-tert-butyl-6-methylphenyl)-3-[(1-ethylpyrrolidin-3-yl)methyl]urea
4-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]azetidin-3-yl}morpholine
2-[2-fluoro-3-(trifluoromethyl)phenyl]-N,6-dimethylpyrimidin-4-amine
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
N-{1-[7-(5-acetylthiophene-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}acetamide
8-[2-(2-hydroxyethoxy)ethyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(1-aminocyclobutanecarbonyl)-N-[2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidine
(4aR,8aR)-2-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-(2-methoxyethyl)-1-[1-(2-methylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
ethyl 2-[3-(2-carbamoylethyl)piperidin-1-yl]-1,3-oxazole-4-carboxylate
(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
(1S,5R)-3-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}-4-methoxyphenol
1-[1-(1,3-benzothiazol-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(naphthalene-1-carbonyl)piperidine
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-{[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino}propanamide
{[(3S,4R)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
1-{5-[1-cyclohexyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}ethan-1-one
6-ethyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-2-methylquinoline-4-carboxamide
5-(1-methylpyrrolidin-2-yl)-3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
4-(1H-pyrazol-1-yl)-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylic acid