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4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1,4-oxazepan-6-ol
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-[3-(2-methoxyacetamido)-2-methylphenyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
1-(piperidin-3-ylmethyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
2-(4-acetylphenoxy)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
4-[(2-aminopyrimidin-5-yl)methyl]-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,9aR)-2,3-dimethyl-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-cyclopentyl-5-[4-(dimethylamino)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
14-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-6-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
6-(cyclopentylamino)-N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]pyridine-3-carboxamide
2-[2-(ethylamino)pyrimidin-5-yl]-N,N,5,7-tetramethylquinoline-4-carboxamide
(3R,4R)-1-[(2-methoxypyrimidin-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
3-(3-hydroxy-3-methylbutyl)-N-[2-(2-methylpiperidin-1-yl)ethyl]benzamide
2-[1-(3-phenylpropyl)-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-2-methoxyphenol
5-[bis(prop-2-en-1-yl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-({[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
9-(pyridin-4-ylmethyl)-3-oxa-9-azaspiro[5.5]undecane
6-({3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)-3-phenylpyrazolo[1,5-a]pyrimidine
2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-N-[2-(2-methoxyphenyl)ethyl]quinazolin-4-amine
3-{[1-(6-chloropyridazin-3-yl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-(3-{[(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)carbamoyl]amino}phenyl)acetamide
9-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
{1-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
(3R,4S)-4-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
1-{[3-(morpholine-4-carbonyl)-1,2-oxazol-5-yl]methyl}-1H-1,3-benzodiazole
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
4-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
4-[4-(ethanesulfonyl)piperazin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
1-cyclopropyl-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-{2-[4-(2-phenylethyl)morpholin-3-yl]acetamido}benzamide
4-methoxy-2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}pyridine
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-hydroxyethyl)benzamide
[2-ethoxy-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenyl]methanol
2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
1-(2-chloropyridin-3-yl)-3-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}urea
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[2-(dimethylamino)ethyl]-4-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyrrolidin-2-one
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
N-(2,3-dimethylphenyl)-N'-[2-(2-ethoxyphenyl)ethyl]propanediamide
6-phenyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide