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1-cyclopentyl-5-oxo-N-[3-(trimethyl-1H-pyrazol-1-yl)propyl]pyrrolidine-3-carboxamide
4-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]pyridine-2-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(2-cyclopropylacetyl)-decahydro-1,6-naphthyridin-2-one
2-[2-(methoxymethyl)pyrimidin-5-yl]-N,7,8-trimethyl-N-propylquinoline-4-carboxamide
2-(2,5-dimethylphenyl)-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
7-methoxy-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3,4,5-tetrahydro-1H-3-benzazepine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]benzamide
4-(benzyloxy)-N-methyl-N-(quinolin-5-ylmethyl)butanamide
2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyridine-3-carboxylic acid
2-{2-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1-propylpiperidin-2-one
N-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}imidazo[1,2-a]pyridine-6-carboxamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[3-oxo-3-(pyrrolidin-1-yl)propyl]amino}methyl)piperidin-2-one
2-ethyl-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
2-(dimethylamino)-7-(3-methyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-ethyl-1-[2-(morpholin-4-yl)-2-oxoethyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(aminomethyl)-4-(2,5-dimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,5-dimethylphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)pyridazine-4-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-hydroxy-2-phenylethyl)-N-methyl-1H-pyrazole-4-carboxamide
2-[(6-methoxypyrimidin-4-yl)amino]-N-(2-methylphenyl)acetamide
1,4-dimethyl-2-(3-phenylpiperazine-1-carbonyl)-1H-indole
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(2-methoxyphenyl)propyl]-1-(propan-2-yl)piperidin-4-amine
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
1-[(2,6-difluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-{3-[1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(4-methylquinolin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methylacetamide
N-(1,4-dioxan-2-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[(3-chloro-5-fluorophenyl)methyl]-2-(methoxymethyl)piperidine
4-benzyl-3-ethyl-1-(propane-1-sulfonyl)-1,4-diazepan-5-one
(3R,5S)-5-(3-fluorophenoxymethyl)-N-[(4-methoxyphenyl)methyl]piperidine-3-carboxamide
N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-methyl-5-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
4-(methylamino)-N-(2-phenoxyphenyl)piperidine-1-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
methyl 4-({[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)carbamoyl}amino)-3-methylbenzoate
3-methyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(4aS,8aR)-6-[2-(propan-2-ylsulfanyl)acetyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(ethanesulfonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-[2-(4-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-pyrazol-1-yl)ethyl]morpholine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
4-(hydroxymethyl)-1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-4-ol
2-amino-6-(3-hydroxyphenyl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
2-(4-methyl-1,4-diazepan-1-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-4-(thiophen-2-yl)butan-1-one
1-{1-[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide