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4-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]-1,4-diazepane-1-carbaldehyde
5-[(1-methylpyrrolidin-2-yl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(5-phenyl-1,2-oxazol-3-yl)formamido]acetic acid
5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrrole-3-carbonitrile
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
2-(3-{1-[3-(pyridin-3-yl)propyl]-1H-pyrazol-3-yl}phenyl)pyridine-4-carbonitrile
3-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}benzoic acid
3-(3-chlorobenzoyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
8-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(2-cyclopropylquinolin-4-yl)methyl](methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
N-ethyl-4-(4-methylphenoxy)-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
1-(3,5-difluorobenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}thiomorpholine-4-carboxamide
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)azepane
3-(3-methoxyphenyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
2-[2-(3-fluorophenyl)piperidin-1-yl]acetamide
(2S,4S)-4-amino-N-methyl-1-[4-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
2-(2-methyl-3-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}-1H-indol-1-yl)acetamide
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-3-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
3-chloro-N-[3-(1H-imidazol-1-yl)propyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
N4-(1H-imidazol-2-ylmethyl)-N4,6-dimethyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
3-fluoro-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]imidazo[1,2-a]pyridine-2-carboxamide
2-methoxy-3-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
6-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
7-methyl-3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,2-dihydroquinolin-2-one
N-cyclopentyl-N'-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}butanediamide
5-chloro-3-fluoro-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
3-phenyl-5-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
(1S,5R)-1,3,3-trimethyl-6-(3-propyl-1H-pyrazole-5-carbonyl)-6-azabicyclo[3.2.1]octane
2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-4-phenylpiperazine
2-amino-4-(3-chloro-5-fluorophenyl)-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(methylamino)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-thiazole-4-carboxamide
4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-one
3-ethyl-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine-3-carboxylic acid
methyl 4-{[3-(2-methoxyacetamido)phenyl]carbamoyl}piperazine-1-carboxylate
7-(5-chloro-3-methyl-1H-indole-2-carbonyl)-1-oxa-7-azaspiro[3.5]nonane
{1-[4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}(pyridin-3-yl)methanol
3-{1-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-2-yl}pyridine
N-(2-fluorophenyl)-5-{[(furan-2-ylmethyl)(methyl)amino]methyl}-1,3-thiazol-2-amine
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]amine
3-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}-1-(3-methylpiperidin-1-yl)propan-1-one
2-({4-phenyl-5-[(trimethyl-1H-pyrazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
2-{2-[1-(4-cyanobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-{5-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}propanamide
N-cyclopropyl-6-methyl-2-oxo-4-(pyridin-3-yl)-N-(1,3-thiazol-5-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenoxy)acetamide