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[(8-methoxy-2H-chromen-3-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-cyclopropyl-1-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(2-methyl-1H-imidazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
6-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
6-methoxy-2-[3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]-1H-indole
(1R,3S)-3-ethoxy-7-(1H-1,2,4-triazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
2-(5-methyl-1H-pyrazol-1-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
(4aS,8aR)-1-(3-aminopropyl)-6-[(3-methyl-1H-indol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N,5-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carboxamide
4,4,4-trifluoro-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}butan-1-one
2-amino-4-phenyl-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
methyl 2-{1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]pyrrolidin-3-yl}acetate
N-(propan-2-yl)-1-[2-(4-{1-[3-(trifluoromethyl)phenyl]propan-2-yl}piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(1-ethylpiperidine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-({[1-(2-fluorophenyl)piperidin-4-yl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
3-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
3,5-dimethoxy-N-{[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]methyl}benzamide
4-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1,4-oxazepan-6-ol
(3aS,7aR)-2-[4-(4-fluorophenyl)butanoyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
9-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-(pyrazin-2-ylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
(3R)-1-{2-amino-7-[(2R)-oxolane-2-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
3-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
methyl[2-(oxan-2-yl)ethyl]({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)amine
N-{1-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide
N-benzyl-N,1-dimethyl-5-({[3-(trifluoromethyl)phenyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-{[3-(2-aminoethyl)phenyl]methyl}-1-(3,5-dimethylphenyl)piperazin-2-one
3-butyl-4-(6-ethyl-2-methylquinoline-4-carbonyl)-1-methylpiperazin-2-one
2-[3,5-dimethyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
2-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4R)-1-(2-ethoxybenzoyl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-(4-ethyl-1H-pyrazol-5-yl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
2-[({1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}oxy)methyl]pyridine
1-[(3-ethenylphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(trifluoromethyl)pyrimidin-2-amine
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]propanamide
4-methyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-[4-(1H-indol-2-yl)phenyl]-1-(oxan-4-yl)piperidine-4-carboxamide
2-methyl-4-oxo-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-5-methyl-1,3-oxazole-4-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
5-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]-N-ethylpyrimidin-2-amine
(4aS,8aR)-1-[(2-aminopyridin-3-yl)methyl]-6-(cyclobutylmethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-({1-[2-chloro-5-(piperidin-1-yl)benzoyl]piperidin-4-yl}methyl)acetamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-[3-(methylsulfanyl)propanoyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one