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N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
11-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4-(2-phenylethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[1-(3-chloro-5-methoxybenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
3,6-dimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
[(3R,4R)-1-(2-phenoxybenzoyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
N-(1-hydroxybutan-2-yl)-2-(2-methoxyphenyl)-N-(thiophen-3-ylmethyl)acetamide
1-{2-hydroxy-3-[2-methoxy-4-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
(3S,4R)-1-(3-chloro-1H-indole-2-carbonyl)-4-methylpiperidine-3,4-diol
2-[3-(2-fluorophenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
(1S,5R)-6-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(difluoromethyl)-N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
2-(4-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}morpholin-3-yl)acetamide
2-(4-chloro-2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
1-methyl-N-[2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidin-4-amine
(1R,3S,5S)-8-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
3-{4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propane-1,2-diol
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
4-(azocan-1-yl)-N,5-dimethyl-N-(oxolan-3-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3,5-dimethyl-2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-indole
7-(4-chloro-3-fluorobenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-10-oxo-N-[4-(pyridin-3-yloxy)phenyl]-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
3,3,3-trifluoro-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)propanamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)(quinolin-6-ylmethyl)amine
2,7-dimethyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
3-(2-fluorophenyl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-phenylpropanamide
8-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3,4-difluorophenyl)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-amine
5-(3-fluorophenoxymethyl)-N-[(1S)-2-hydroxy-1-phenylethyl]-1H-pyrazole-3-carboxamide
{1-[(1-benzyl-1H-imidazol-5-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
N-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-2,3-dimethoxybenzamide
2-(4-methylpentyl)-4-(thiophene-3-sulfonyl)morpholine
methyl (1R,3S,3aR,6aS)-3-[2-(2-methoxyethyl)pyrimidin-5-yl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]benzamide
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-benzyl-8-(5-methoxyfuran-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
(3S)-1-(2,1,3-benzoxadiazole-5-carbonyl)-N,N-dimethylazepan-3-amine
N,3-dimethyl-2-oxo-1-(2-phenylethyl)-N-propyl-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-6-methylpyridazine
(2R,3R)-3-amino-1'-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(6-methoxypyridin-3-yl)-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[2-(2-fluorophenyl)-1-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-4-(5-methylfuran-2-yl)benzamide
5-(4-benzylpiperidine-1-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-(piperidin-1-yl)butanamide
2-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
3-[5-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-(propan-2-yl)propanamide
2-methyl-8-(4-phenoxybutanoyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one