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N-methyl-5-({[(5-methylfuran-2-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]pyrazine-2-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-4-ol
1-(2-methylpiperidin-1-yl)-2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethane-1,2-dione
N-(3,5-dimethylphenyl)-4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
ethyl 4-(7-chloro-3-{[N-cyclopropyl-1-(2-oxo-1,2,5,6,7,8-hexahydroquinolin-3-yl)formamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
2-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
6-ethyl-4-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)-2H-chromen-2-one
1-(cyclopropylmethyl)-N-ethyl-5-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethyl-N-(1-hydroxybutan-2-yl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
1-(1-{4-[(benzylcarbamoyl)methyl]phenyl}piperidin-4-yl)piperidine-3-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)pyrrolidine-3-carboxylic acid
3-(1-methylpiperidin-2-yl)-1-[4-(9H-purin-6-yl)piperazin-1-yl]propan-1-one
(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1,4-oxazepan-6-yl)methanol
1-[3-(1H-1,2,4-triazol-5-yl)benzoyl]piperidine-3-carbonitrile
N-{[(2S,4S)-4-fluoro-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl]methyl}ethane-1-sulfonamide
6-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
5-(1-cyclopropanecarbonylpyrrolidin-2-yl)-N-[2-(pyridin-3-yloxy)ethyl]thiophene-2-carboxamide
7-methyl-3-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2-dihydroquinolin-2-one
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3R,4R)-4-(hydroxymethyl)-1-(2,4,5-trimethoxybenzoyl)piperidin-3-ol
N-[2-(3-chlorophenyl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-6-methylpyridine-3-carboxylic acid
1-(4,5-dimethylthiophene-2-carbonyl)-4-methyl-1,4-diazepan-6-ol
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-methylthiophene-2-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
4-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-1-oxaspiro[4.4]nonan-2-one
3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
N-(2,3-dihydroxypropyl)-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
(2S,4S)-4-amino-N-ethyl-1-(naphthalene-2-sulfonyl)pyrrolidine-2-carboxamide
4-cyclobutyl-N-[(1-ethylpiperidin-2-yl)methyl]-6-methylpyrimidin-2-amine
2-[2-(4-fluorophenoxy)ethyl]-N-(propan-2-yl)benzamide
(4aR,8aR)-2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
ethyl 4-[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]piperidine-1-carboxylate
9-[(4-methoxy-3-methylphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
4-{[1-(carbamoylmethyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-[4-(butan-2-yl)phenyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carboxamide
5-(2-fluorophenoxymethyl)-N-(2-hydroxy-2-phenylethyl)-1H-pyrazole-3-carboxamide
(2S)-2-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxypropanamide
(4aS,7aR)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-fluoro-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
(4aS,7aR)-1-(4-methylpyrimidine-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylimidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(cyclopropylmethyl)-5-({[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}amino)azepan-2-one