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1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]urea
2-(benzyloxy)-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]ethan-1-one
1-(difluoromethyl)-N-[1-(3-methoxyphenyl)ethyl]-N-methyl-1H-pyrazole-5-carboxamide
N-cyclopropyl-2-(dimethylamino)-2-(4-methylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
2,6-dimethoxy-N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)pyridine-3-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[3-(thiophen-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
methyl 2-[8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-[(4-chlorophenyl)methyl]-N-(3-cyclopentylpropyl)-6-oxopiperidine-3-carboxamide
2-(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)-N-(propan-2-yl)acetamide
9-{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,5R)-6-(cyclobutylmethyl)-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
1-(6-{3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridin-3-yl)ethan-1-one
2-{3-methyl-5-[4-(morpholine-4-carbonyl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
2-{1-[(2-fluorophenyl)methyl]-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
(3S,4S)-4-(propan-2-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]pyrrolidine-3-carboxylic acid
3-{1-[2-(3-ethyl-1H-pyrazol-5-yl)-1H-imidazol-1-yl]ethyl}adamantan-1-ol
2-oxo-N-[2-(pyridin-2-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-cyclopropyl-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-2-[(phenylsulfanyl)methyl]pyrimidin-4-ol
4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(5-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-2-(propan-2-yloxy)phenyl)methanol
2-[3-(2-methoxyethyl)-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]-1-methylpiperidine
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-[2-(pyrazin-2-yl)ethyl]acetamide
6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
9-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3,4-dichlorophenyl)-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}morpholine
4-acetamido-N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}benzamide
1-(4-{[(2R,5S)-5-[(3-ethoxyphenyl)methyl]oxolan-2-yl]methyl}piperazin-1-yl)ethan-1-one
ethyl 4-{[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]amino}piperidine-1-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-ethyl-2-methylpyrimidin-4-amine
1-[(benzylcarbamoyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
8-[(1S,3R)-3-aminocyclopentanecarbonyl]-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1R,3R)-3-aminocyclopentyl]-1-ethyl-5-methyl-1H-pyrazole-3-carboxamide
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-phenylbutane-1,2-dione
methyl 3-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]benzoate
2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[(propan-2-yl)amino]pyridine-3-carboxamide
2-(1H-pyrazol-1-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]butanamide
2-{1-[(1-pentylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
1-(2-methoxyethyl)-4-{4-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl}pyrrolidin-2-one
2-(5-methyl-1,3-oxazole-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-(furan-2-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenylpropanamide
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyridine-2-carboxamide
(1S,6R)-9-(4-phenyl-1,3-thiazol-2-yl)-3,9-diazabicyclo[4.2.1]nonan-4-one
1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}imidazolidin-2-one
4-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3,3-dimethylpiperazin-2-one
N-methyl-3-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
N3-{3-[(furan-2-ylmethyl)sulfanyl]propyl}piperidine-1,3-dicarboxamide