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N,N-dimethyl-3-(4-phenoxybenzoyl)piperidine-1-sulfonamide
methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})(pyrrolidin-3-ylmethyl)amine
4-(pyridin-3-ylmethoxy)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
N-(2,3-dihydro-1H-inden-4-yl)-2-(2-hydroxyethyl)piperidine-1-carboxamide
N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
2-[(isoquinolin-5-yloxy)methyl]-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
N-methyl-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-2-carboxamide
[1-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidin-2-yl]methanamine
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
1-[1-(methylsulfanyl)propan-2-yl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
5-ethanesulfonamido-1-methyl-2-phenyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
1-(4-benzylpiperidin-1-yl)-3-[1-(thiophene-3-carbonyl)piperidin-4-yl]propan-1-one
1-[(4-fluorophenyl)methyl]-4-(5-methoxyfuran-2-carbonyl)-1,4-diazepane
3-[(6-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)methyl]-N-methyl-1,2,4-oxadiazole-5-carboxamide
3-[1-(2,5-dimethoxyphenyl)-1H-imidazol-2-yl]-7-fluoro-1,2-dihydroquinolin-2-one
5,6-dimethyl-2-[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]-1H-1,3-benzodiazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
9-(2-amino-6-methylpyrimidin-4-yl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-[(dimethylcarbamoyl)amino]-N-(pyridin-3-ylmethyl)acetamide
3-(2-chlorophenyl)-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2-methoxyethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3-methoxyphenyl)methyl]-N-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-3-amine
propyl 4-(2,3-dihydro-1H-inden-2-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
4-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1-cyclohexylpiperazin-2-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-(pyrrolidin-3-yl)benzamide
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}[(6-methylpyridin-2-yl)methyl]amine
N-ethyl-5-methyl-6-(4-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(5S,9aS,9bS)-5-(4-chlorophenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-hydroxy-4-methoxy-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]benzamide
2-amino-7-(2-cyclopentyl-2-phenylacetyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(3,4-dimethoxyphenyl)-2-methyl-2,8-diazaspiro[4.5]decane-8-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperazin-1-yl)-1-(pyrrolidin-1-yl)ethan-1-one
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-3-(1H-1,2,4-triazol-1-yl)propanamide
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methylimidazolidin-2-one
3-{4-[1-(3-chloro-2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(pyrazin-2-yl)acetamide
(4aS,7aR)-1-[2-oxo-2-(piperidin-1-yl)ethyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperazine-1-carboxylate
1-benzyl-N3-cyclopropyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(2-methyl-1,3-thiazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-butyl-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
{3-[(2-fluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
4-{1-[1-(thiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-2-yl}pyridine
(3R,4S)-1-(4-chloro-3-methyl-1H-pyrazole-5-carbonyl)-4-cyclopropylpyrrolidin-3-amine
2-(1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole