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4-(1-methanesulfonylpyrrolidine-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
3-[5-(1-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,4-oxadiazol-3-yl]pyridine
4-(4-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
8-(1H-imidazol-2-ylmethyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[1-(2-fluorobenzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
1-[(4aR,8aR)-7-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
3-[(1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
methyl 2-methyl-2,8-diazaspiro[4.5]decane-8-carboxylate
4-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-6-(methoxymethyl)pyrimidine
N-(1,3-dihydroxypropan-2-yl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-(3-hydroxypropyl)-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-[2-(1H-indol-3-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
(4aS,8aR)-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(5-methylthiophene-2-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-(1-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)pent-4-enamide
3-hydroxy-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
1-(3-aminoazepan-1-yl)-2-(2H-1,2,3-benzotriazol-2-yl)ethan-1-one
4-{1-benzyl-5-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
5-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
4-(2,4-dioxoimidazolidin-1-yl)-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]benzamide
6-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
(2R)-2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-4-methylpentanamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-3-yl)piperazin-1-yl]ethan-1-one
3-[(3R,4S)-1-(3-chloro-2-methylbenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(2-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-methyl-5-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]pyrimidin-4-ol
N5,N5-dimethyl-N6-[(3-methylphenyl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-N-methylpiperidine-2-carboxamide
6-methyl-N-{2-[1-(pyridin-2-ylmethyl)piperidin-3-yl]ethyl}pyridine-3-carboxamide
N-[2-(2-oxopyrrolidin-1-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
4-[1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]benzoic acid
3-benzyl-5-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,2,4-oxadiazole
3-[1-(2-phenylethyl)piperidin-4-yl]-1,3-oxazolidin-2-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(1-methylpyrrolidin-3-yl)amino]pyridine-3-carboxamide
{5-[1-(2,2-diphenylethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
1'-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
(1S,4S)-2-(2-fluorophenyl)-5-(quinoxalin-6-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[2-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(2-fluorophenoxy)piperidine
2-{1-[2-(4-methoxynaphthalen-1-yl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
3-(1-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-3,4-dihydroquinazolin-4-one
4-(3-methoxyphenyl)-3,3-dimethyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperazine-1-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3S,4R)-1-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N'-(2,5-dimethylphenyl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)propanediamide