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(2R,3R,6R)-5-(6-methylpyridazin-3-yl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-benzyl-N-methyl{[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]amino}sulfonamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2,6-dimethoxybenzamide
1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-amine
2-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxo-N-(1,3-thiazol-2-yl)acetamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-3-oxopiperazine-1-carboxamide
(2S,4R)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
1'-(5-phenyl-1,2-oxazole-3-carbonyl)spiro[indene-1,4'-piperidine]
2-(4-fluorophenyl)-1-(furan-2-carbonyl)piperidine
(1S,5R)-6-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{4-[(cyclohexylmethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
9-[(2-ethylpyrimidin-4-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-methylfuran-3-carboxamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
6-(hydroxymethyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-1,4-oxazepane-4-carboxamide
2-[(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)sulfanyl]-6-methyl-3,4-dihydropyrimidin-4-one
N-[(3S,4R)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-{2-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]propyl}-3-methylpyridine
1-(5-methyl-1,3-oxazole-4-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
N,3-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-propyl-1H-pyrazole-4-carboxamide
N-benzyl-5-(pyridin-4-yl)furan-2-carboxamide
1-{1'-[(2-butyl-1H-imidazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-4-(1H-imidazol-1-yl)butan-1-one
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
4-methyl-N-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
3-{3-[3-(3-fluoro-4-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
4-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
3-{1-[(4-methylpiperidin-1-yl)sulfonyl]piperidin-3-yl}benzoic acid
[(3S,5R)-1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
5-(2,6-dimethylphenoxymethyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
3-(5-{2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
3-(3-methoxypropyl)-1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]piperidine-3-carboxylic acid
6-(azepan-1-yl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(4aS,8aR)-1-butyl-6-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(1-phenylcyclohexanecarbonyl)-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
1-[(3-methoxyphenyl)methyl]-N-[3-(methylsulfanyl)propyl]-6-oxopiperidine-3-carboxamide
4-[1-(2-hydroxyethyl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
N-[(2,5-dimethoxyphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
1-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
2-[1-(2H-1,3-benzodioxol-5-yl)-5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-3-yl]acetamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-(dimethyl-1,2-oxazol-4-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-5-methyl-1,3-oxazole-4-carboxamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide