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8-(2,2-diphenylacetyl)-1,8-diazaspiro[4.5]decan-2-one
3-{[4-methyl-3-(2-oxoimidazolidin-1-yl)phenyl]formamido}-N-(1,3-thiazol-2-yl)propanamide
5-methyl-1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(butan-2-yl)-5-{2-[(pyridin-4-ylmethyl)amino]ethyl}pyrrolidin-2-one
2-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]phenoxy}-N,N-dimethylacetamide
3-(prop-2-en-1-yl)-1-[3-(thiophen-2-yl)propanoyl]piperidine-3-carboxylic acid
(3R,4S)-3,4-dimethyl-1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-ol
1-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidine-4-carbonitrile
4-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}benzoic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-hydroxy-N-methyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,2-oxazole-5-carboxamide
4-(3-hydroxypyrrolidine-1-carbonyl)-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-[(4-fluorophenyl)methyl]-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-{[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}quinolin-7-ol
(3R,4S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
5-(hydroxymethyl)-4-{[4-(3-hydroxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methylpyridin-3-ol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
(2S,4S)-4-({[3-(benzyloxy)phenyl]methyl}amino)-1-[(3-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
1-({4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
2-(2-aminoethyl)-N-[1-(4-methanesulfonylphenyl)ethyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
2-[3-(morpholin-4-ylmethyl)phenyl]quinoline
2-cyclopentyl-1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-{3-[(diethylamino)methyl]phenyl}-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-2,4-dimethylpyrimidine
3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-3-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)acetamide
3-[(4-methanesulfonylpiperazin-1-yl)methyl]-8-methyl-2-(thiophen-2-yl)quinoline
2-ethyl-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}butan-1-one
(2R,3R)-3-amino-1'-(1-phenylcyclopropanecarbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[3-(2-propyl-1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
[(2S)-1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}pyrrolidin-2-yl]methanol
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
3-[(3R,4S)-1-[2-(2-chlorophenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]ethane-1-sulfonamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(5-methylpyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)propanamide
N3-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]piperidine-1,3-dicarboxamide
(1R,7S)-6-(3-oxopiperazine-1-carbonyl)-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
(1R,5S,8R)-3-[(2,3-difluoro-6-methoxyphenyl)methyl]-8-methoxy-3-azabicyclo[3.2.1]octane
(1S,5R)-6-benzyl-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
2-(2,3-dimethoxyphenyl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
4-(1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}azetidin-3-yl)morpholine
N3-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-{4-[(pyridin-2-yl)amino]piperidin-1-yl}propan-1-one