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1-methyl-2-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-indole
2-[3-({methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)piperidin-1-yl]ethan-1-ol
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-2,7-naphthyridin-4a-ol
4-methyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrimidine
1-(4-chloro-1-ethyl-1H-pyrazole-3-carbonyl)-3-phenylpiperazine
4-fluoro-2-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}phenol
N,N-dimethyl-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(2-oxoazepan-3-yl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-(2-methoxyethyl)-4-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
3-amino-N-[3,5-difluoro-4-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide
2-[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-N-(2-methylphenyl)acetamide
1-{[4-(methylsulfanyl)phenyl]methyl}-3-(pyrrolidin-1-yl)pyrrolidine
1-[3-(2-oxopyrrolidin-1-yl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
(furan-2-ylmethyl)(quinolin-4-ylmethyl)(thiophen-3-ylmethyl)amine
1-(4-{[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]methyl}thiophen-2-yl)ethan-1-one
3-[5-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-2-methyl-6-(trifluoromethyl)pyridine
2-(3-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
N-(2-chlorophenyl)-3-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
1-(cyclopropylmethyl)-3-hydroxy-3-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]piperidin-2-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
3-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-4-fluorobenzene-1-sulfonamide
3-[3-(ethoxymethyl)-5-[(pyrimidin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
5-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-ylmethyl]-2-ethoxypyridine
(1R,3S)-3-(2-aminoethoxy)-7-(6-methylpyridine-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(3S,4S)-1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
1-[1-(4-methylpentanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2,4-dimethoxy-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
[2-(dimethylamino)ethyl](methyl)(2-{[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]oxy}hex-5-en-1-yl)amine
1-butyl-4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-2-one
3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}propanamide
(1S)-2-phenyl-1-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethan-1-amine
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
4-ethyl-N,N-dimethyl-6-(4-{[1-(6-methylpyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)pyrimidin-2-amine
3-(4-chlorophenyl)-4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]butanoic acid
({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
(2S)-2-amino-N-[(3-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-3-(1,3-thiazol-4-yl)propanamide
4-(furan-2-ylmethyl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-methylphenyl)-1-{2-[(2,3,4-trimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
(2R)-2-amino-1-[4-(2-chlorophenoxy)piperidin-1-yl]-3-methoxypropan-1-one
1-(1-methyl-1H-indole-2-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
2-(4-{[4-(benzyloxy)-2-methoxyphenyl]methyl}morpholin-3-yl)-N,N-dimethylacetamide
1-ethyl-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-2-{2-[(1-propanoylpiperidin-3-yl)formamido]ethyl}-1,3-thiazole-5-carboxylic acid
N-(2-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
2-methyl-5-(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one