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5-ethyl-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
(3aR,6aR)-2-cyclopentyl-5-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](1H-imidazol-4-ylmethyl)methylamine
N-ethyl-N-methyl-2-{[1-(thiomorpholin-4-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
3-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
(3R,4S)-4-(4-methoxyphenyl)-1-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)pyrrolidin-3-amine
1-(2-methylphenyl)-3-[2-(methylsulfanyl)ethyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
6,6-dimethyl-5-oxo-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}thiomorpholine-3-carboxamide
N,5-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-2-yl}propan-1-ol
N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-[1-(pyridin-3-yl)propan-2-yl]-6-azaspiro[2.5]octane-1-carboxamide
1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-phenylethane-1,2-dione
(2S)-2-({4-[ethyl(2-methylprop-2-en-1-yl)amino]-5-methylthieno[2,3-d]pyrimidin-6-yl}formamido)-3-phenylpropanamide
N4-methyl-N4-[3-(oxolan-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-(4-fluorophenyl)-4-[6-(methoxymethyl)pyrimidin-4-yl]morpholine
4-(1H-indole-6-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-{[1-(4-fluorophenyl)pyrrolidin-3-yl]methyl}-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-N,N-dimethylaniline
9-(2-methoxypyridine-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[(4-ethylphenyl)methyl]-1,4-diazepan-5-one
1,3-dimethyl-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-methylpropyl)benzamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
[2,4,6-trimethyl-3-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)phenyl]methanol
3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazine
[1-(oxan-4-ylmethyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
1-ethyl-N-[(2-methyl-1,3-oxazol-4-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
1-[2-(morpholin-4-yl)-2-oxoethyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(azepane-4-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-({[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)propan-1-ol
5-{5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
5-methyl-3-[3-(2,3,4-trimethoxyphenyl)phenyl]-1,2,4-oxadiazole
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
4-(azepan-1-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyridine-2-carboxamide
2-ethyl-4-(oxolan-2-ylmethyl)-1-(propan-2-yl)piperazine
8-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-2-(2-{methyl[(3-methylpyridin-2-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
N-[4-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)phenyl]acetamide
4-(3-methylbutyl)-11-[(pyridin-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(3R,4S)-4-({[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)oxolan-3-ol
(1S,5R)-3-(5-methyl-1,3,4-oxadiazol-2-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenylacetamide
(1H-imidazol-4-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine