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N-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methanol
9-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-6-oxa-9-azaspiro[4.5]decane
N-butyl-2-[methyl({5-methylpyrazolo[1,5-a]pyrimidin-7-yl})amino]acetamide
N-ethyl-2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}acetamide
2-[4-(3-methyl-1H-pyrazole-5-carbonyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
dimethyl({[4-methyl-5-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
2-(ethoxymethyl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}pyrrolidine
N-[2-(2-chloro-6-methylphenoxy)ethyl]-1,4-dithiepan-6-amine
N-[2-(ethanesulfonyl)ethyl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
methyl 2-(N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamido)acetate
3-chloro-6-[4-(oxan-4-yl)piperazin-1-yl]pyridazine
3-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}methyl)pyrrolidin-3-ol
N-(1-methyl-1H-indazol-5-yl)-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
2-[3-(2-methylpropyl)-5-[phenyl(1H-1,2,3,4-tetrazol-1-yl)methyl]-1H-1,2,4-triazol-1-yl]pyridine
2-cyclopropanecarbonyl-8-[(2,4,6-trimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(3,4-dimethylphenyl)-1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-amine
5-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]-2-methoxypyridine
(3aS,7aR)-5-methyl-2-[2-(2-methylphenyl)benzoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-(2-hydroxyethyl)-7-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1-benzofuran-2-carboxamide
1-cyclopentyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-5-oxopyrrolidine-3-carboxamide
N-ethyl-1-methyl-N-(2-methylprop-2-en-1-yl)-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
4-(4-chlorophenoxy)-1-(1H-pyrrole-3-carbonyl)piperidine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-benzyl-3-(2-fluoro-6-methoxyphenyl)-N,N-dimethyl-1H-1,2,4-triazol-5-amine
5-cyclopropanecarbonyl-1'-{[4-(methylsulfanyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(4,6-dimethylquinolin-2-yl)sulfanyl]-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propan-1-one
5-methanesulfonyl-4-(piperidin-3-yl)-N-(piperidin-4-ylmethyl)pyrimidin-2-amine
1-cyclobutanecarbonyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
(4aS,7aR)-1-(2-ethoxyacetyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetamido)phenyl]pentanamide
4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-1,2,3-triazole
(1S,5R)-6-benzyl-3-[2-(pyridin-4-ylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]propanamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-(4-chlorophenyl)-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclobutane-1-carboxamide
3-[(methylamino)methyl]-4-[(2-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({5-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-[(oxan-4-yl)amino]pyridine-3-carboxamide
2-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)quinolin-4-ol
2-amino-6-cyclobutyl-4-[3-(1H-pyrazol-1-ylmethyl)phenyl]pyridine-3-carbonitrile
3-(butan-2-yl)-1-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
1-(furan-2-ylmethyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
2-(3-methoxypropyl)-9-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]cyclopropane-1-carboxamide
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyridin-2-ol
4-(1H-imidazol-1-yl)-1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]piperidine-4-carboxylic acid