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(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-acetamido-2-methylpropanoyl)pyrrolidine-3-carboxylic acid
3-cyclopentaneamido-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
2-cyclopropyl-N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
N-[(2-fluorophenyl)methyl]-3-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-3-yl}propanamide
5-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]pyrimidine-2,4-diol
methyl 2-(1-{3-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-5-(pyrrolidine-1-sulfonyl)phenyl}-N-methylformamido)acetate
4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
[(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
[(3S,7S)-5-[4-(dimethylamino)benzoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
1-(4-ethylpiperazin-1-yl)-3-{1-[2-(pyridin-3-yloxy)acetyl]piperidin-4-yl}propan-1-one
N-[2-(3-methoxyphenoxy)ethyl]-N-methyl-4-(piperidin-3-yl)benzamide
dimethyl({2-[3-(morpholin-4-ylmethyl)phenoxy]phenyl}methyl)amine
2-[4-(2-aminopyrimidin-4-yl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butan-1-one
5-methoxy-4-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,4-dihydropyridine-2-carboxamide
ethyl 1-(cyclopropylmethyl)-5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(2-chlorophenyl)-3-{1-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
ethyl 2-[1-(2-phenylpyrimidine-5-carbonyl)piperidin-2-yl]acetate
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1,3-thiazol-2-yl)-decahydro-1,6-naphthyridin-2-one
N-{2-[(pyridin-3-yl)amino]ethyl}-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
6-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,6R,8aS)-2-(5-ethyl-1,2,4-oxadiazol-3-yl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-fluoro-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-5-sulfamoylbenzamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-{2-[(5-fluoroquinazolin-4-yl)amino]ethyl}methanesulfonamide
N-[3-(pyridin-4-yl)propyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(2,4-difluorophenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-methylthiophene-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[2-(benzylsulfanyl)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-phenyl-8-[3-(pyridin-3-yl)propanoyl]-1,8-diazaspiro[4.5]decan-2-one
5-[6-(aminomethyl)pyridin-3-yl]-N,N-diethylfuran-2-carboxamide
7-(cyclopropylmethyl)-2-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-(1-ethyl-1H-imidazol-2-yl)-1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(3-methoxy-4-methylbenzoyl)piperidine
2-(morpholin-3-yl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethan-1-one
4-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
3-(2-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N,3-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]-1,2-oxazole-5-carboxamide
3-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
(1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperidin-2-yl)methanamine
1-(1-{[4-(2-aminoethyl)phenyl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
1-{4-[2-methoxy-4-(4-phenylpiperazine-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
2-[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-(1,2-oxazinan-2-yl)propanamide