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[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-(1-phenylcyclopentanecarbonyl)pyrrolidin-3-yl]methanol
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(thiophen-2-yl)propanamide
(1S,5R)-6-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
3-(2,5-dioxoimidazolidin-4-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
2-{9-[3-(4-methylphenyl)propanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amine
2-cycloheptanecarbonyl-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
6-(oxolane-2-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-methyl-2-{4-[(4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}acetamide
3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]urea
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-methylthiophene-3-carbonyl)piperidine
2-(5-fluoro-2-methylphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-(4-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-4-oxobutyl)acetamide
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}benzamide
N,2-dimethyl-N-(2-phenyl-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl)furan-3-carboxamide
methyl(pyrimidin-5-ylmethyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
methyl 3-(5-aminopyrazin-2-yl)benzoate
4-cyclobutyl-2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methylpyrimidine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
2-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
1-[2-ethyl-7-(thiophene-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidine
N-cyclopropyl-3-[5-(quinoxalin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-amine
(3S,5R)-5-(cyclopropylcarbamoyl)-1-(5-fluoropyrimidin-2-yl)piperidine-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyrimidin-2-amine
3-[2-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
2-(pyrimidin-5-yl)-6-(pyrrolidine-1-carbonyl)pyrazine
4-benzyl-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)pyrrolidin-2-one
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(2-phenoxyethyl)piperazine
N,2-dimethyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 4-{[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}butanoate
(5S,9aS,9bS)-5-(3-chlorophenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(6-methyl-2-propylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
6-(hydroxymethyl)-N-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-1,4-oxazepane-4-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
3-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
7-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
(2S,4S)-4-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]pyrrolidine-2-carboxylic acid
N-cyclopropyl-1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
8-{2-[3-(dimethylamino)pyrrolidin-1-yl]acetyl}-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}propanamide
methyl 4-{[(2-{1-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
4-{1-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyridine