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2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-indole
(2S,4R)-4-amino-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-N-methylpyrrolidine-2-carboxamide
3-methyl-8-[4-(pyridin-4-yl)pyrimidin-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methanesulfonylethyl)-5-methylpiperidin-2-one
methyl (2S,4S,5R)-1,2-dimethyl-4-[methyl(pyridin-2-ylmethyl)carbamoyl]-5-(2-methylphenyl)pyrrolidine-2-carboxylate
3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
5-[1-(oxolan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]isoquinoline
N-[(5-methylfuran-2-yl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
N1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}propane-1,3-diamine
2-methyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-acetamidobenzamide
4-[5-(2-acetylphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]piperazin-2-one
1-(1-benzofuran-2-carbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
2-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
N-[1-(methoxymethyl)cyclopentyl]-N'-[2-(propan-2-yl)phenyl]butanediamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-imidazole-5-carboxamide
2-({4-[1-(2-hydroxyethyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]phenyl}(methyl)amino)ethan-1-ol
3-[2-(diethylamino)ethyl]-3H,4H-pyrido[4,3-d]pyrimidin-4-one
N-benzyl-3-[(1-cyclobutylpiperidin-4-yl)oxy]benzamide
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(pyridin-2-yl)acetamide
3-ethyl-8-(2-phenoxybenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
(3R,9aR)-3-(propan-2-yl)-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(2-methylquinolin-5-yl)pyrimidin-2-amine
3,5-dichloro-4-methyl-N-[2-(methylsulfamoyl)ethyl]benzamide
N-ethyl-N-[(2-fluorophenyl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-3-yl}-2-phenylethan-1-one
2-methyl-5-{4-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
N-[2-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
5-(2-ethyl-6-methylpyrimidin-4-yl)-1H-indole
N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
1-methyl-4-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)piperazine-2-carboxylic acid
1-cyclopropanecarbonyl-4-[4-(2-methylpiperidine-1-carbonyl)phenoxy]piperidine
3-(5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-1-(2-phenylphenyl)piperazin-2-one
N-methyl-3-{2-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]phenyl}propanamide
3-methyl-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
ethyl 4-(3-phenylpropyl)-1-(thiophene-2-carbonyl)piperidine-4-carboxylate
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(thiophen-3-yl)acetic acid
2-{[(4-methoxynaphthalen-1-yl)methyl](methyl)amino}-N,N-dimethylpropanamide
1-{2-[(4-methylphenyl)sulfanyl]ethyl}-3-[2-(oxolan-2-ylmethoxy)phenyl]urea
N-(2-methoxyethyl)-2-oxo-7-propoxy-N-(thiophen-2-ylmethyl)-2H-chromene-3-carboxamide
5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]quinoxaline
1-methyl-1'-(9H-purin-6-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N,N-dimethyl-2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide