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1-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
1-methyl-N-(2-phenylethyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methoxy-6-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)-N,N-bis(propan-2-yl)benzamide
1-[2-(piperazin-1-yl)ethyl]-N-[3-(pyridin-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(5-chloro-1H-indol-2-yl)methyl]acetamide
3-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
N,4,6-trimethyl-2-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
4-hydroxy-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(4-fluorophenyl)-4-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]butane-1,4-dione
2-(4-acetyl-1,4-diazepan-1-yl)-2-(3-ethylphenyl)acetic acid
2-benzyl-9-(3-methylbut-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-hydroxy-N-({1-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
(1s,4s)-4-[2-(4-phenylpiperidin-1-yl)acetamido]cyclohexane-1-carboxylic acid
N-benzyl-5-cyclopropyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-oxazole-4-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-(4-oxo-4-phenylbutyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-[1,2,4]triazolo[4,3-a]pyrimidine-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-2-one
N-{2-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamido]-4-methylphenyl}pentanamide
1-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-1,4-dihydroquinolin-4-one
3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1-[2-(pyrrolidin-1-yl)ethyl]-1,2-dihydroquinolin-2-one
2-(1-{5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-cyclopropyl-5-(1H-imidazol-4-ylmethyl)-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-(pyrrolidin-3-yl)-3-{[3-(1H-1,2,4-triazol-1-yl)propyl]sulfamoyl}benzamide
4-{4-[(4-fluorophenyl)methyl]piperazin-1-yl}-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
5-{[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]methyl}-3-methyl-1,2-oxazole
(1R,3S)-3-(2-aminoethoxy)-7-(5-chloro-2-fluorobenzoyl)-7-azaspiro[3.5]nonan-1-ol
4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-2-one
N-[(4-fluorophenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
dimethyl[2-({[5-(oxolan-2-yl)thiophen-2-yl]methyl}(thiophen-3-ylmethyl)amino)ethyl]amine
N-(2-methoxyethyl)-3-(5-methylfuran-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
(1R,5S)-6-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
8-chloro-2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]quinoline
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-N-(dimethyl-1H-1,2,4-triazol-3-yl)benzamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
8-[2-(2-methylphenyl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
2-[3-(propan-2-yl)-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]pyridine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-5-methylphenol
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(furan-2-yl)-2-oxoacetamide
N-cyclopropyl-1-{1-[5-(hydroxymethyl)furan-2-carbonyl]piperidin-4-yl}piperidine-3-carboxamide
N,2,3,5-tetramethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N,N-diethyl-5,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
3-[(2-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
1-(oxolan-3-ylmethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide