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N-methyl-2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[1-(3-methylpyridin-2-yl)propyl]-1H-1,3-benzodiazole-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(2-phenylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-(benzyloxy)-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propan-2-ol
3-({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,3-oxazolidin-2-one
N-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
1-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)propanamide
dimethyl({1-[1-(2-methylbutyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
3-methyl-1-propyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-pyrazole-4-carboxamide
1,1-dioxo-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
3-(3-aminoazepan-1-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-benzoyl-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-[(3-methylphenyl)methyl]piperazin-2-one
(3R,4R)-1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N4-(furan-3-ylmethyl)-N4-methyl-6-(morpholin-4-yl)pyrimidine-2,4-diamine
(1R,2R,6S,7S)-4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
[(2,5-dimethoxyphenyl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[(2,3-dimethoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}benzoic acid
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
4-chloro-N-cyclohexyl-N-[(4-fluorophenyl)methyl]-1-methyl-1H-pyrazole-3-carboxamide
2-(2,4-dichlorophenoxy)-1-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]ethan-1-one
5-(2,6-dimethoxyphenyl)-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]acetamide
3-[(2R,3R,6R)-5-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-(4-chloro-1H-pyrazol-1-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
1-[2-(1H-indol-4-yl)pyrimidin-4-yl]pyrrolidin-3-ol
7-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
methyl 6-{6-oxo-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}pyridine-2-carboxylate
(1R,2S,3R,4R,5S)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}tricyclo[3.2.1.02,4]octane-3-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
{5-[(E)-2-phenylethenyl]-1H-1,3-benzodiazol-2-yl}methanol
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(oxolan-3-ylmethyl)-1H-pyrazole-3-carboxamide
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{5-[5-(oxolan-2-yl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(1-methylpyrrolidin-3-yl)quinoline-4-carboxamide
1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-methyl-2-({2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}amino)-3,4-dihydropyrimidin-4-one
5-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethoxy-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
5-amino-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-phenyl-1H-pyrazole-3-carboxamide
1-(cyclopropylmethyl)-5-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3aR,6aR)-2-(cyclobutylmethyl)-5-(3,4-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-hydroxy-4-methylpentan-1-one
2-benzyl-N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-thiazole-4-carboxamide
8-cyclopropanecarbonyl-2-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid