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N,N-diethyl-4-(1H-imidazol-1-yl)aniline
N-[(3R,4S)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-propylpyrrolidin-3-yl]oxane-4-carboxamide
5-(2,4-dimethoxyphenyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,2,4-triazin-3-amine
3-(2-ethyl-1H-imidazol-1-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
4-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)pyridine
ethyl 1-(1H-1,3-benzodiazol-2-ylmethyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
1-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)-1H-1,3-benzodiazole-5-carboxamide
1-{2-[3-(4-chlorophenyl)piperidin-1-yl]-2-oxoethyl}-4-ethylpiperazine-2,3-dione
5-[(1-carbamoylcycloheptyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(1H-indol-3-yl)butanamide
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-{2-[1-(4-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}azepan-2-one
1-[5-(2-methylpropyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-6-phenyl-2,3-dihydropyridazin-3-one
1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-(1-ethyl-1H-imidazol-2-yl)-1-[3-(2-fluorophenyl)benzoyl]piperidine
2,6-dimethoxy-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine
3-[benzyl(1H-imidazol-2-ylmethyl)amino]-1λ6-thiolane-1,1-dione
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-{1-[(3E)-pent-3-enoyl]pyrrolidin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]thiophene-2-carboxamide
3-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
[(3R,4R)-1-(1-benzothiophen-2-ylmethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-(dimethylamino)ethyl]-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-{5-[2-(2,4-difluorophenyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methylacetamide
4-[4-(2-methoxyethoxy)piperidin-1-yl]-6-methylpyrimidin-2-amine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3,5-dimethyl-1-[1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)azetidin-3-yl]-1H-pyrazole
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-(4-fluorophenyl)-5-[3-(pyrrolidin-1-yl)propyl]-1,2,4-oxadiazole
N-[(2-methylphenyl)methyl]-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-(cyclopropylmethyl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
8-[3-(furan-2-yl)-4-phenylbutanoyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
1-cyclohexyl-3-methyl-4-[(1s,4s)-4-aminocyclohexyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
2-(4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl)pyridine
2-(2-methoxyethyl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,3-benzoxazole-6-carboxamide
7-propyl-3-(pyridin-2-yl)-2,4,5,7-tetraazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
6-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl 2-(2-benzyl-3-oxopiperazine-1-carbonyl)benzoate
4-(1H-imidazol-1-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidine-4-carboxylic acid
6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
8-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,4R)-1-[4-(4-fluorophenyl)butanoyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-(2-{[1-(4-phenylphenyl)piperidin-4-yl]amino}ethyl)-1,3-oxazolidin-2-one