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5-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
2-{5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-(cyclopropylmethyl)-7-[1-(propan-2-yl)piperidine-3-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{3-[4-(1H-imidazol-2-yl)phenoxy]propyl}dimethylamine
(1S,6R)-3-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-(2-methoxyethyl)-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-(thiophen-3-ylmethyl)acetamide
2-(4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperidin-1-yl)acetamide
8-(5-acetylpyridin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyridin-3-yl)propan-1-one
(5S,9aS,9bS)-2-cyclopentyl-5-(7-methoxy-2H-1,3-benzodioxol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane-1-carbaldehyde
[(3R,4R)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)quinolin-7-ol
2-cyclopropyl-5-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]pyrimidin-4-ol
3-[3-(trifluoromethyl)benzoyl]piperidine
N,3,6-trimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
8-chloro-2-{[4-(dimethylamino)azepan-1-yl]methyl}-1,4-dihydroquinolin-4-one
2-(1H-indol-3-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3S)-3-({5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)azepan-2-one
1-{2-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenyl}ethan-1-one
N-[2-(2,3-dichlorophenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,3-oxazolidin-2-one
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-benzotriazole
4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}pyrrolidine-1-sulfonamide
4-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-oxobutane-1-sulfonamide
methyl 5-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-6-methyl-1,2-dihydroquinolin-2-one
2-[(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
(3R,4S)-4-(4-methoxyphenyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-amine
5-(2,6-difluorophenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
1-cyclopentyl-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-(adamantan-1-ylmethyl)-N-methyl-5-(phenoxymethyl)-1,2-oxazole-3-carboxamide
2-methyl-2-(2-{[(1-methylpiperidin-2-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
3-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-4H-chromen-4-one
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
N,6-dimethyl-4-oxo-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-dihydropyridine-3-carboxamide
N-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
2-(butylsulfanyl)-6-(4-methanesulfonylpiperazin-1-yl)pyrimidin-4-amine
1-({1-[3-amino-3-(3,4-dimethoxyphenyl)propanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
8-methoxy-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[2-chloro-4-(pyrrolidine-1-carbonyl)phenoxy]-1-methanesulfonylpiperidine
methyl (2R,4S)-4-hydroxy-1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidine-2-carboxylate
N-methyl-5-[4-(1H-pyrazol-3-yl)benzoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
5-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
benzyl({[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})(2-phenylethyl)amine
(3aR,6aR)-2-benzyl-5-[2-(3-fluorophenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(tert-butylsulfamoyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]benzamide
4-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazine-1-sulfonamide