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1-(2,5-difluorobenzoyl)-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-methyl-6-(propan-2-yl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1R,5R)-6-(cyclopropylmethyl)-3-(3,6-dimethylpyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(4aR,7aS)-1-(cyclopropylmethyl)-4-{2-[4-(propan-2-yl)phenyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(3R,4R)-1-(3-ethoxybenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-{[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}piperidine
2-tert-butyl-6-[1-(4-methylphenyl)cyclopropanecarbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1,5-dimethyl-4-{[methyl(quinolin-5-ylmethyl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-[(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
N-(oxan-4-yl)-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
N-({5-[(3-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-(2-hydroxypropyl)-9-(pyrrolidine-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
3-butyl-4-ethyl-1-[2-oxo-2-(3-phenylpiperazin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-methyl-2-(morpholin-4-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
1-benzyl-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
[(3-chloro-5-fluorophenyl)methyl](1H-imidazol-2-ylmethyl)methylamine
2,6-dichloro-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
dimethyl({4-[2-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1,3-thiazol-2-yl}methyl)amine
2-methyl-4-[4-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)phenyl]but-3-yn-2-ol
4-(1-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)thiomorpholine
(1S,5R)-3-cyclobutanecarbonyl-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(3-methoxyphenyl)piperazine
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
2-(2-ethoxypyridin-3-yl)-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-(2,1,3-benzoxadiazol-5-ylmethyl)acetamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[3-(trifluoromethyl)phenyl]acetamide
2-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
N-cyclohexyl-3-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)propanamide
N-(pyridin-2-ylmethyl)-1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
2-(1-benzoylpiperidin-4-yl)-1,2,3,4-tetrahydroisoquinolin-4-ol
N-(2,5-dimethylphenyl)-3-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]propanamide
2-({methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)quinolin-8-ol
2-(3-chloro-4-hydroxyphenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-[3-(3-fluorophenyl)phenyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxamide
7-(2-cyclohexylethyl)-2-methanesulfonyl-2,7-diazaspiro[4.5]decan-6-one
N-cyclopentyl-3-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1,2-oxazole-5-carboxamide
N-(3,5-dimethoxyphenyl)-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}propanamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-phenyl-1,2-oxazole-5-carboxamide
1-methyl-N-[(3-methylphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-[3-fluoro-5-(propan-2-yloxy)phenyl]-N,N-dimethylpyridazin-3-amine
4-cyclopentyl-N-[4-(2-oxopyrrolidin-1-yl)phenyl]-1,4-diazepane-1-carboxamide
(1s,4s)-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-hydroxy-N-methylcyclohexane-1-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(1H-pyrrol-1-yl)propanoyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(pyridin-2-yl)propan-1-one
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide