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4-(oxan-4-yl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(piperidin-4-ylmethyl)benzamide
3-methyl-8-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}-N-[(3R)-pyrrolidin-3-yl]benzamide
1-{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}-4-propylpiperazine
1-cyclohexyl-3-methyl-5-(oxan-4-yl)-1H,4H-pyrazolo[3,4-d]imidazole
N-(4-{4-[(oxan-4-ylmethyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
5-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]pyridine-3-carboxamide
1-(4-chlorobenzoyl)-3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
N-benzyl-5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
2-[2-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)phenoxy]acetic acid
4-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]benzamide
3-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-(2,3-dimethylphenyl)urea
(2S,3R)-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-N-(prop-2-en-1-yl)bicyclo[2.2.1]heptane-2-carboxamide
1-(6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]pyrrolidine-2-carboxylate
5-[7-(2-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]-N-methylfuran-2-carboxamide
(1S,5R)-N-(3-methoxyphenyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-[cyclohexyl(methyl)amino]-3-[3-({[(3-methyloxetan-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N,1-dimethyl-5-oxo-N-[(4-phenoxyphenyl)methyl]pyrrolidine-3-carboxamide
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(1H-pyrazol-3-ylmethyl)acetamide
1-ethyl-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine-3-carboxamide
2-{[(4-cyanophenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{[(5-methoxypyrimidin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
2-methyl-5-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1H-1,3-benzodiazole
3-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}-5-methyl-1,2-oxazole
4-{3-[4-(1H-pyrazol-5-yl)phenyl]phenyl}-4H-1,2,4-triazole
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperazine-2-carboxylic acid
1-(3,5-difluorophenyl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-{1-[(5-tert-butyl-2-hydroxyphenyl)methyl]piperidin-4-yl}piperidin-3-ol
3-{[(1-benzothiophen-2-ylmethyl)amino]methyl}-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
4-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)(3-phenylpropyl)amine
(4aS,8aS)-2-[4-(4-propylphenyl)benzoyl]-decahydro-2,7-naphthyridin-4a-ol
5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-N-(1H-1,2,4-triazol-3-ylmethyl)piperidine-3-carboxamide
3-{1-[(2-aminopyrimidin-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxybenzoyl)piperidine
2-butyl-8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]amino}adamantan-1-ol
(3S,9R)-11-(4-ethylbenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
(1S,5R)-6-methyl-3-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-2-oxo-N-[3-(1H-pyrazol-1-yl)phenyl]-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
4-(5-ethoxyfuran-2-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
methyl 3-({pyrazolo[1,5-a]pyrimidin-2-ylformamido}methyl)-5-(thiophene-2-sulfonamido)benzoate
4-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]benzoic acid