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(2S)-2-amino-3-(1H-indol-3-yl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]ethan-1-ol
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-{2-[(3S,4S)-4-{[(dimethylcarbamoyl)amino]methyl}-3-hydroxypiperidin-1-yl]-2-oxoethyl}benzamide
6-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,4-diazepan-5-one
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrrolidin-2-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
(2S,4R)-1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-N,N-diethyl-4-propanamidopyrrolidine-2-carboxamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine
(2S)-2-[5-(2-ethylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]-2-phenylethan-1-ol
3-(3-hydroxyquinoxalin-2-yl)-1-{octahydropyrrolo[1,2-a]piperazin-2-yl}propan-1-one
2-{2-[methyl(pyridin-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-2-yl)piperazine
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}ethan-1-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)-N-(propan-2-yl)benzamide
N-(2-methylpropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-cyclopentyl-4-[(2-fluoro-4-methoxyphenyl)methyl]-1,4-diazepane
N2-(5-ethylpyrimidin-2-yl)-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
2-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}pyridine-4-carboxamide
N-(2H-1,3-benzodioxol-4-ylmethyl)-1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[2-(3-methoxypropyl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-5-[(2-ethyl-4-methyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(methylamino)pyridine-4-carboxamide
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-5-(pyrrolidine-1-carbonyl)pyridine
4-methyl-N-[(3R,5S)-1-(3-methylbut-2-en-1-yl)-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
5-{3-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-4-methylphenyl}-1H-1,2,3,4-tetrazole
3-methoxy-1-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
N-(4-hydroxybutan-2-yl)-4-{methyl[(methylcarbamoyl)methyl]sulfamoyl}benzamide
7-(cyclobutylmethyl)-2-[(3-hydroxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{1-[(2-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}piperidin-4-ol
4-(1,3-thiazol-2-yl)-1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazole
2-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}benzoic acid
3-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}pyrrolidin-3-ol
1-ethyl-3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2,5-dimethyl-1H-pyrrole
(2S,3R)-2-{[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-3-hydroxybutanamide
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
methyl 4-{[(4aR,8aS)-1-(1,2,3-thiadiazole-4-carbonyl)-decahydro-1,6-naphthyridin-6-yl]methyl}benzoate
4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-[2-(trifluoromethoxy)benzenesulfonyl]piperidine
methyl 5-[(1-methoxy-1-oxopropan-2-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2,6-dimethoxypyridin-3-yl)-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]morpholine-4-carboxamide
4-{[1-(4-methoxyphenyl)-5-(5-methyl-1,2-oxazol-4-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2-benzyl-9-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-3,4-dihydroquinazolin-4-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[3-(dimethylcarbamoyl)-5-{[(4-phenylbutan-2-yl)amino]methyl}phenyl]pyridine-2-carboxamide