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3-ethyl-6-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
(1S,5R)-3-(3-propyl-1H-pyrazole-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclobutanecarbonyl-N-(1H-indol-6-ylmethyl)piperidine-4-carboxamide
N-[(5-methylfuran-2-yl)methyl]-7-oxo-2-propanamido-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-cyclopentyl-N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)acetamide
1-benzyl-8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-2-methyl-N-(thiophen-3-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
1-(4-chlorophenyl)-N-[1-(pyridin-2-yl)propan-2-yl]cyclobutane-1-carboxamide
7-(2-methyl-4-phenylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
5-acetamido-1-ethyl-N-(furan-2-ylmethyl)-2-(3-methoxyphenyl)-N-(prop-2-yn-1-yl)-1H-1,3-benzodiazole-7-carboxamide
5-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
1-(4-oxo-4H-chromen-6-yl)-3-[(2S)-oxolan-2-ylmethyl]urea
N-{1-oxaspiro[4.4]nonan-3-yl}-2-propyl-1,3-thiazole-4-carboxamide
2-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}-2-(2,4,6-trimethylphenyl)acetic acid
8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(3S,9aR)-8-(2,5-difluorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[5-(6-chloro-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]acetamide
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyridine-3-carboxylic acid
N-cyclopropyl-4-(3-fluorophenyl)-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}benzamide
3-({[1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
4-[(3-chloro-1-benzothiophen-2-yl)methyl]-4H-1,2,4-triazole
5-{[benzyl(methyl)amino]methyl}-N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
(2R)-1-[(5-chloro-2,4-dimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
6-[5-(methoxymethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(2-aminoethyl)-2-methyl-N-[2-(morpholin-4-yl)ethyl]pyrimidin-4-amine
3-{3-[1-(pyrrolidin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}quinoline
2-[2-({[2-hydroxy-3-(4-methylphenoxy)propyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
1-(2-fluorophenyl)-4-[1-(thiophen-2-ylmethyl)piperidin-3-yl]piperazine
3-[1-(butan-2-yl)-1H-pyrazol-5-yl]-1-[2-(4-methoxyphenyl)ethyl]urea
2-{[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}benzonitrile
3-{4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperazin-1-yl}pyrazine-2-carbonitrile
1-(benzyloxy)-8-[2-(pyridin-3-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
5-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-1H-pyrazole-3-carboxamide
8-{[2-(2-hydroxyethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-3-ol
2-ethoxy-5-{2-[(thiolan-3-yl)amino]pyrimidin-4-yl}benzoic acid
2-ethyl-4-methyl-N-[(1R,2S)-2-phenylcyclopropyl]-1,3-oxazole-5-carboxamide
1-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
3-[5-(2,2-dimethyloxan-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
2-ethyl-8-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
3-{2-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[(3R,4S)-4-cyclopropyl-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl]cyclopropanesulfonamide
ethyl 2-[1-(3-hydroxypyridine-2-carbonyl)piperidin-2-yl]acetate
3-(3-methylphenyl)-1-(4-methylphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
2-amino-6-cyclobutyl-4-(2,3-dimethoxyphenyl)pyridine-3-carbonitrile
[(3R,4R)-4-[(dimethylamino)methyl]-1-[5-(1H-indol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-yl]methanol
(1R,3S)-7-[(2-chlorophenyl)methyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-{4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperazin-1-yl}-2-phenoxyethan-1-one
2-[4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]pyrazine
(2S,3S)-2-amino-3-methyl-1-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pentan-1-one