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8-methyl-3-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}-2-(thiophen-2-yl)quinoline
N-[2-(benzyloxy)phenyl]-1-oxa-7-azaspiro[3.5]nonane-7-carboxamide
(2R,3R)-3-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-benzyl-4-(3-cyanopyridin-2-yl)piperazine-1-sulfonamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(methylsulfanyl)phenyl]urea
2-(2,3-dimethoxyphenyl)-1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazole
N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-3-(1H-pyrazol-4-yl)benzamide
2-(3-hydroxyadamantan-1-yl)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
3-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
methyl (2S,4R)-4-(dimethylamino)-1-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]pyrrolidine-2-carboxylate
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
1-(3-chlorophenyl)-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine
{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}(pyridin-4-ylmethyl)amine
2-(2-oxopiperidin-1-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}acetamide
5-acetyl-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)thiophene-3-carboxamide
4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenol
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-(trifluoromethyl)benzene-1-sulfonamide
2-cyclopentyl-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(1-{1-[1-(4-methylphenyl)piperidin-4-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(pyridin-4-yl)acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-fluorobenzoyl)-2,8-diazaspiro[4.5]decan-3-one
[(3R,4R)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-ethyl-N-(2-methoxyethyl)acetamide
2-amino-4-(cyclohex-3-en-1-yl)-6-(1,3-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-(1,4-dioxan-2-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-(2H-1,3-benzodioxol-5-yl)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]piperidin-3-amine
3-[3-(propan-2-yloxy)benzoyl]piperidine
2-ethyl-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-[2-oxo-2-(piperazin-1-yl)ethyl]acetamide
(4aS,7aR)-1-(butane-1-sulfonyl)-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(dimethylamino)oxan-4-yl]methyl}-4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(1-methylpiperidin-3-yl)-N-(pyridin-4-ylmethyl)propanamide
2-benzyl-4-(2-methoxy-5-methylbenzenesulfonyl)morpholine
5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-2-(pyridin-3-yl)pyrimidin-4-ol
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-[(2R,3R)-2-methoxy-1'-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
2-[(1S,5R)-3-[2-(3,4-dimethylphenoxy)ethyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-(5-aminopyridin-3-yl)-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
methyl N-{2-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-oxoethyl}carbamate
N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-({[6,7-dimethoxy-4-(piperidin-1-yl)quinazolin-2-yl]methyl}(2-hydroxyethyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
2-{2-[cyclopentyl(methyl)amino]ethyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
{3-ethyl-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}methanol
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(8-fluoroquinoline-2-carbonyl)pyrrolidin-3-yl]methanol
1-(cyclohexylmethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(4-{[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]methoxy}phenyl)ethan-1-one
methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine