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1-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N,3,6,7-tetramethyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-benzofuran-2-carboxamide
(3S)-3-({5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)azepan-2-one
3-methyl-7-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-[(dimethylamino)methyl]-N-[2-(4-fluorobenzenesulfonyl)ethyl]furan-2-carboxamide
methyl 5-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-5-oxopentanoate
4-[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-[1-(2-fluorophenyl)propan-2-yl]-1-(morpholin-4-ylmethyl)cyclopentan-1-amine
6-[1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[2-(3-methyl-1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,5-difluoropyridine-2-carboxamide
2-{[5-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
4-chloro-1-methyl-3-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
(3S,4S)-4-propyl-1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidine-3-carboxylic acid
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]acetamide
3-(1-methyl-1H-pyrazol-4-yl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
3-[4-fluoro-3-(hydroxymethyl)phenyl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
(2,1,3-benzoxadiazol-5-ylmethyl)[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
5-fluoro-4-(morpholin-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyrimidin-2-amine
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4H-1,2,4-triazole
6-[2-(cyclohex-1-en-1-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[3-(2-fluorophenyl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
(2R)-2-amino-3-methoxy-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}propanamide
3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-methyl-3,4-dihydroquinazolin-4-one
(2E)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)-3-(thiophen-2-yl)prop-2-enamide
N-(2-fluoro-5-methylphenyl)-3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carboxamide
2-[1-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethan-1-ol
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2-{2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{5-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-2-methylphenyl}imidazolidin-2-one
N-[3-(methylsulfanyl)propyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
8-(butan-2-yl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1-methyl-1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[(3R,4S)-1-(3-phenoxypropanoyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
8-(pent-2-yn-1-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}-3-methylbutan-1-ol
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
N-cyclopropyl-2-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)pyridine-4-carboxamide
1-[3-(furan-2-yl)phenyl]-3-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
1-(8-methylquinolin-5-yl)-3-[3-(methylsulfanyl)propyl]urea
3-{4-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperazin-1-yl}pyrazine-2-carbonitrile
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
N3-cyclooctyl-N5-(1-methoxypropan-2-yl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
1-({2-methoxy-5-[1-(2-methylpropyl)-4-phenyl-1H-imidazol-5-yl]phenyl}methyl)-1H-1,2,4-triazole
4,6-dimethyl-5-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)-2H-pyran-2-one
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(1H-indol-3-yl)ethyl]acetamide