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5-(dimethylamino)-2-(2-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
6-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
5-{[3-(1-methylpiperidin-2-yl)propanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(2-chlorophenyl)-4-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperazin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-2-oxo-8-(pyrimidin-2-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
(3aR,6aR)-2-acetyl-5-[(1-benzyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3aS,6aS)-2-cyclobutanecarbonyl-5-(6-cyclopropylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-4-hydroxy-3-methylbenzamide
6-(3-ethylpiperazin-1-yl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-(4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
N-{1-[1-(dimethylsulfamoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
2-[methyl({4-methyl-5-[1-(5-methylpyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methylphenyl)ethan-1-one
6-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}-1-phenylethan-1-ol
N-{[(3S,4S)-3-hydroxy-1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl]methyl}morpholine-4-carboxamide
(4aS,8aR)-1-propyl-6-(quinoline-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(2-methylphenyl)methyl]-N-(propan-2-yl)acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
(2E)-1-[(2R,3R)-2-hydroxy-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-methylbut-2-en-1-one
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-6-(pyridin-4-yl)-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
4-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methylbenzamide
3-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-(3-methoxyphenyl)urea
N-(1-ethyl-1H-pyrazol-5-yl)-3-{[3-(N-methylacetamido)pyrrolidin-1-yl]methyl}benzamide
5-(4-acetylpiperazine-1-carbonyl)-6-methyl-4-(2-phenylethyl)-1,2,3,4-tetrahydropyrimidin-2-one
(1R,3S,5S)-8-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-8-azabicyclo[3.2.1]octan-3-ol
{1-[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
(2S)-2-(methoxymethyl)-N-[3-(1,3-thiazol-4-yl)phenyl]pyrrolidine-1-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
6-(2-chlorophenyl)-N-cyclobutyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-yl]methanesulfonamide
2-[4-(4-methoxyphenyl)butan-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1,5-dimethyl-4-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-(carbamoylmethyl)-N-{[1-(2-fluorophenyl)cyclopentyl]methyl}piperidine-4-carboxamide
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-(2-chlorophenyl)propan-1-one
5-methoxy-2-(3-methyl-3-phenylpiperidine-1-carbonyl)-4H-pyran-4-one
2-methoxy-6-{2-[(3-methylpyridin-4-yl)amino]ethyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-methyl-2-{[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]amino}acetamide
2-ethyl-8-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(2-fluoro-6-methoxybenzoyl)-4-phenylpiperidin-4-yl]ethan-1-one
N-{2-[2-(3-fluorophenyl)piperidin-1-yl]-2-oxoethyl}benzamide
4-ethyl-3-({1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-amino-N-methyl-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxamide
2-(morpholin-4-yl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-2-(pyridin-3-yl)acetamide