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5-amino-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1H-pyrazole-3-carboxamide
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
(2S,4S)-N-ethyl-4-[3-(3-fluorophenyl)benzamido]-1-methylpyrrolidine-2-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-N-(4-ethylphenyl)propanamide
5-methyl-4-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}thiophene-3-carboxamide
(3S)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine-3-carboxylic acid
4-ethyl-3-[1-(isoquinolin-5-ylmethyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(5-phenyl-1H-pyrrole-2-carbonyl)-3-(1H-pyrazol-5-yl)piperidine
1-[(1-acetylpiperidin-4-yl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
4-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}thiomorpholine
5-(furan-2-yl)-1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
1-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
3-(4-carbamoyl-3-chlorophenyl)-4-methylbenzamide
2-methyl-5-[2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(pyridin-3-yl)propanamide
N-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-3-methoxybenzamide
2-(4-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}morpholin-3-yl)acetic acid
2-{4-[2-(3-fluorophenoxy)acetyl]-2-oxopiperazin-1-yl}benzonitrile
1-cycloheptyl-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
1-(2-aminoethyl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-{4-[4-(methylamino)pyrimidin-2-yl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
8-methoxy-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
N-(2-methoxyethyl)-1-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-(pyridin-4-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidin-2-amine
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
6-butyl-2-(4-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-ylmethyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[(2E)-3-(3-chlorophenyl)prop-2-enoyl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
8-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(2E)-3-(4-chlorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]prop-2-en-1-one
4-[2-(3,5-difluorophenyl)-1H-imidazol-1-yl]benzene-1-sulfonamide
5-{5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]methylamine
4-{[5-(5-ethyl-1,3,4-thiadiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,4-oxazepane
2-(butylsulfanyl)-6-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]pyrimidin-4-amine
(3S,4R)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-fluoro-5-methanesulfonamidophenyl)urea
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
1-ethyl-6-oxo-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}piperidine-3-carboxamide
4-[2-(N-ethylpropanamido)-4-methylphenoxy]thiane-4-carboxylic acid
N-(2,3-dihydroxypropyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
2-amino-4-[2-(ethylamino)pyrimidin-5-yl]-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
(1S,5R)-3-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[1-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-4-yl]-7-fluoro-N,N-dimethylquinoline-4-carboxamide
6-fluoro-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
2-(butylsulfanyl)-5-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)pyrimidine
(2-{2-[1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine