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1-(1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
2-(3-methoxypropyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
8-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-3-methyl-2H,3H,5H,6H,7H,8H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
1-[(2-chloro-6-fluorophenyl)methyl]-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-ethyl-1H-1,2,4-triazole
2-[(3,4-difluorophenyl)methyl]-8-(oxolane-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-(3-chloro-4-methoxyphenyl)-2,4-dimethyl-1,3-thiazole
3-(1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
7-(cyclopropylmethyl)-2-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(2,3-dimethylphenyl)-N-[(3-ethoxy-4-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1,3-thiazol-2-yl)piperidin-4-yl]propanamide
5-ethyl-4-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)-2-methylpyrimidine
[(3R,4R)-1-[3-(difluoromethoxy)benzoyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
methyl 5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
4-({[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl](methyl)amino}methyl)-1-cyclopentylpyrrolidin-2-one
3-(2,6-dimethylphenoxy)-1-(oxane-4-carbonyl)azetidine
2-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-N,6-dimethylpyrimidin-4-amine
1-(4-aminopyrimidin-2-yl)-4-(3-methylphenoxy)piperidine-4-carboxylic acid
(3S)-N-tert-butyl-2-[6-(hydroxymethyl)pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[2-(2-ethylpyrimidin-5-yl)-8-methylquinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
(3S,4S)-4-cyclopropyl-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(3-methoxyphenoxymethyl)-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N,N-bis(prop-2-en-1-yl)benzamide
5-{[1-(2,4-difluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-dimethylimidazolidine-2,4-dione
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)propanamide
2-ethoxy-4-{[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]methyl}phenol
(3R,4R)-3-cyclopropyl-4-methyl-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}pyrrolidin-3-ol
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
4-ethyl-3-{[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1'-(2H-1,3-benzodioxol-5-ylmethyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
[5-(4-phenyl-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-5-yl)furan-2-yl]methanol
8-(3-hydroxypyridine-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-(6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carbonyl)-1,4-diazepan-5-one
4-hydroxy-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-phenylpyrimidine-5-carboxamide
7-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
1-(2-{3-[(methylsulfanyl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
3-(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-1λ6-thiolane-1,1-dione
(3S,4R)-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
10-methoxy-5-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-(1H-pyrazol-4-yl)benzamide
(3S,4R)-1-[(8-methoxyquinolin-2-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
9-(5-acetylpyridin-2-yl)-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-{[2-hydroxy-5-(pyridin-3-yl)phenyl]methyl}piperidine-2-carboxylate
1-(furan-2-ylmethyl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}piperidine-3-carboxamide
1-ethyl-3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one