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1-({1-[6-(1H-pyrazol-4-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4,4,4-trifluorobutyl)piperidine
2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-(4-fluoro-3-methoxyphenyl)morpholine-4-carboxamide
2-(4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-5-methyl-2-oxopiperazin-1-yl)benzonitrile
2-(2-fluorophenyl)-2-hydroxy-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}acetamide
4-{[2-(2-fluorophenyl)ethyl]amino}-5-methyl-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
ethyl[3-(5-methylfuran-2-yl)butyl][2-(1H-pyrazol-1-yl)ethyl]amine
8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{4-[(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)methyl]phenyl}acetamide
(3aS,6aS)-2-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2-methoxyphenoxy)-1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidine-4-carboxylic acid
5-acetyl-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}acetamide
4-{[1-(3-fluorophenyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
N-[(2-propoxyphenyl)methyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-amino-2-[(E)-2-phenylethenyl]pyrimidine-5-carbonitrile
N-[2-(pyrrolidine-1-sulfonyl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-ethyl-N-[1-(methoxymethyl)cyclopentyl]-1H-pyrazole-4-carboxamide
8-(2-ethylpyrimidine-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
2-(3-hydroxypropyl)-9-[(3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N,2-dimethyl-N-(1,2-oxazol-3-ylmethyl)-3-(1H-pyrazol-1-yl)propanamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
6-[(oxan-4-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-{1-[1-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
2-[2-(dimethylamino)phenyl]-6,7-dimethoxyquinazolin-4-amine
2-({6-[2-(trifluoromethyl)morpholin-4-yl]pyrimidin-4-yl}amino)ethan-1-ol
11-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
1-(cyclopropylmethyl)-N-ethyl-5-[2-(3-methylphenyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethyl-N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
(3R,4S)-1-methanesulfonyl-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)(pyrazin-2-ylmethyl)amine
2-chloro-5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}pyridine
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azocane
3-(3-fluorophenyl)-N-(4-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
1-(cyclopropylmethyl)-3-({[(2,3-difluoro-4-methylphenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
1-[2-(1H-imidazol-4-yl)acetyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4-diazepane-6-carboxylic acid
4-[4-({[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]acetamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]piperazine
1-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-{[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazole
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-({1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}methyl)furan-2-carboxamide
N-[1-(4-methanesulfonylphenyl)ethyl]-3-azaspiro[5.5]undecan-9-amine
(4aR,8aS)-6-cyclopentyl-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one