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1-(2-cyclopentyl-2-phenylacetyl)-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
4-[({[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)methyl]-1-ethylpyrrolidin-2-one
1-methyl-N-[(4-phenylmorpholin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
1-(2-fluorobenzoyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-(1-cycloheptylpiperidin-3-yl)-3-(methylsulfanyl)propanamide
1-{1'-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
7-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-{[(1S)-1-cyclohexyl-2-hydroxyethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
2-(dimethylamino)-N-[5-({[1-(methoxymethyl)cyclopentyl]carbamoyl}amino)-2-methylphenyl]acetamide
3-({1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
2-{5-[2-(dimethylamino)-1,3-thiazol-5-yl]-4-phenyl-1H-imidazol-1-yl}acetic acid
[(3R,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-methyl-1-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azetidin-3-yl}piperidine
1-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]benzamide
2-(2H-1,3-benzodioxol-5-yl)-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}acetic acid
2-{4-[(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}pyridine-4-carbonitrile
1-(oxan-4-yl)-4-(quinoxalin-2-yl)-1,4-diazepan-6-ol
4-(4-fluoro-2-methylphenoxy)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine-4-carboxylic acid
(4aS,8aR)-1-[2-(ethylsulfanyl)ethyl]-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
(2S)-1-{2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carbonyl}pyrrolidine-2-carboxylic acid
(3S)-3-benzyl-4-[(8-chloroquinolin-2-yl)methyl]piperazin-2-one
1'-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
(4aS,7aR)-1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-4-(cyclopropylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,9aR)-3-(hydroxymethyl)-8-{[3-(methylsulfanyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-amine
4-(6-amino-5-methylpyridin-3-yl)-2-chlorobenzamide
1-(1-methyl-1H-imidazol-2-yl)-2-({thieno[2,3-d]pyrimidin-4-yl}amino)ethan-1-ol
3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]phenyl}urea
(3aR,5S,6S,7aS)-5,6-dihydroxy-N-[2-(thiophen-2-yl)ethyl]-octahydro-1H-isoindole-2-carboxamide
{5-methyl-7-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-({2-[4-(1H-pyrazol-1-yl)phenoxy]phenyl}methyl)morpholine
2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
3-(2-methoxyethyl)-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-3-(thiophen-2-ylmethyl)urea
N,N-dimethyl-7-(4-methyl-1H-imidazole-5-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[3-methoxy-4-(pyrrolidin-1-yl)phenyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl})amine
5-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
9-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-amino-6-(2,4-dimethoxyphenyl)-4-(4-hydroxyphenyl)pyridine-3-carbonitrile
3-({1-[(4,5-dimethylfuran-2-yl)methyl]pyrrolidin-3-yl}methyl)-1-phenylurea
1-({1-[1-(cyclopropanesulfonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
3-(4-chloro-1H-pyrazol-1-yl)-1-(3-{[2-(dimethylamino)ethyl](methyl)amino}piperidin-1-yl)propan-1-one
N-(3-cyclopentylpropyl)-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide