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N-ethyl-2-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N'-cyclopentyl-N-(2-methanesulfonamidoethyl)butanediamide
ethyl 4-[6-(pyridin-4-ylmethyl)-6-azaspiro[2.5]octane-1-carbonyl]piperazine-1-carboxylate
3-cyclohexyl-N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1H-pyrazole-4-carboxamide
(3aS,6aS)-2-cyclopentyl-5-[5-(methoxymethyl)thiophene-2-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(oxolan-2-ylmethyl)piperazine
2-[5-(2H-1,3-benzodioxole-5-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2-hydroxyphenyl)ethan-1-one
(2R,4S)-1-(2-chlorobenzenesulfonyl)-4-hydroxypiperidine-2-carboxylic acid
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2,5-dimethylfuran-3-carbonyl)piperidine
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)imidazo[1,2-a]pyridine-3-carboxamide
N-[(3S,4R)-1-(2-methanesulfonylacetyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1-benzofuran-5-carboxamide
methyl 2-[1-(2-methoxyethyl)-2,4-dioxo-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(3R,4R)-4-(azepan-1-yl)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]piperidin-3-ol
(4aR,7aS)-1-acetyl-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 6-(butan-2-yl)-2-{[(4-chlorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[3-(benzyloxy)propyl]-N,N-dimethylbenzamide
2-cyclopentyl-1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-ethoxypropan-1-one
4-(1-methyl-1H-imidazol-2-yl)-1,3-diphenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-1H-pyrazole
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N'1-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropane-1,1-dicarboxamide
4-{1-[4-(6-methylpyridin-3-yl)phenyl]ethyl}morpholine
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-N-ethylpyrrolidine-3-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(pyridin-4-yl)acetamide
5-[({2-amino-3-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}formamido)methyl]-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
2-(4-fluorophenyl)-N-[1-(pyridin-2-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
4-{1-methyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
{4-benzyl-1-[4-(1H-indol-3-yl)butan-2-yl]piperidin-4-yl}methanol
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-methylphenyl)benzamide
1-[3-({3-[3-(methoxymethyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-(2-hydroxyphenoxy)acetamide
[(2S,6S)-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-cyclopropanecarbonyl-1'-(6-methylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3S,4R)-1-[(8-fluoroquinolin-2-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}naphthalen-2-ol
3-{[butyl(methyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(2-{methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
N-cycloheptyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-1-(1,3,4-thiadiazol-2-yl)urea
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-3-(piperidin-4-ylmethyl)benzamide
1-{[1-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid