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N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-2,3-dihydro-1H-isoindole
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(3-sulfamoylphenyl)urea
3-ethyl-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperazine
4-[(dimethylamino)methyl]-1-(5-methylpyridine-3-carbonyl)azepan-4-ol
ethyl 1-[5,8-dimethoxy-3-({[(3S)-2-oxoazepan-3-yl]amino}methyl)quinolin-2-yl]piperidine-4-carboxylate
4-hydroxy-2-(4-methylphenyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]pyrimidine-5-carboxamide
6-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-[1-(4-methyl-1,3-thiazol-2-yl)piperidin-3-yl]-1H-1,3-benzodiazole
N-cyclopropyl-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]furan-3-carboxamide
2-[(dimethylcarbamoyl)amino]-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
1-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propylurea
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-(hydroxymethyl)-1-[(4-phenoxyphenyl)methyl]azepan-4-ol
2-(3-chlorophenoxy)-1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
2-(cyclopropylmethyl)-9-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-fluorophenyl)-N-methyl-N-(thiophen-3-ylmethyl)oxane-4-carboxamide
1-(2-fluorophenyl)-4-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}piperazine
8-fluoro-3-(1-propylpiperidin-4-yl)-3,4-dihydroquinazolin-4-one
5-[({[3-(2-{4-[4-(3-fluorophenyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
4-hydroxy-3-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
[(2-fluorophenyl)methyl](methyl){[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}amine
4-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}pyridine
5-[(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)methyl]-1H-indole
2-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[(2-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(4-methylpiperazin-1-yl)ethyl]-6-phenylpyridazin-3-amine
7-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-{4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}piperidine-1-carboxamide
(3R,4R)-4-ethyl-1-[4-(furan-2-yl)benzoyl]piperidine-3,4-diol
ethyl 4-[(4-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
1-[1-(2,5-dimethoxyphenyl)ethyl]-5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazole
N-{3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-2-phenylacetamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(1R,2R,6S,7S)-4-(2,3-dihydro-1H-isoindole-1-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
3-(1H-pyrazol-1-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
3-(ethoxymethyl)-5-(1-methylcyclopropyl)-1-(2-phenylethyl)-1H-1,2,4-triazole
1-(2-methoxyacetyl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
3-(2H-1,3-benzodioxol-5-yl)-5-(cyclopropylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}but-3-en-1-one
7-(6-chloro-1,3-benzothiazol-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
methyl 4-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-1-yl)benzoate
N-(3-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}-3-oxopropyl)methanesulfonamide
4-(1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid
5-ethyl-5-{3-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
(1R,2R,6S,7S)-4-[5-(morpholine-4-carbonyl)pyridin-2-yl]-4-azatricyclo[5.2.1.02,6]decane
[(4-{[(3S)-3-ethylmorpholin-4-yl]sulfonyl}phenyl)sulfamoyl]dimethylamine
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidin-4-amine
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-5-carboxamide