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5-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-(4-methanesulfonylphenyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
2-{4-[(3,5-dimethylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-[1-(pyrazin-2-yl)piperidin-3-yl]urea
4-benzyl-N-(1-propyl-1H-1,3-benzodiazol-5-yl)piperazine-1-carboxamide
5-[5-(5-cyclopropyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(2H-1,2,3-benzotriazol-2-yl)-1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
4-(4-methoxyphenyl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}butan-1-one
5-chloro-N-[2-(1H-indol-1-yl)ethyl]-N-methylpyridine-2-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-[2-(1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
7-fluoro-2-methyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]quinoline
4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5,6-dimethyl-2-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
1-({1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-2-methyl-4-(2-methylphenyl)piperazine
1-cyclopentyl-4-oxo-N-(prop-2-en-1-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
(1S,5R)-6-[(3,4-dichlorophenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,5S)-3-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-3,4-dimethyl-5-sulfamoylbenzamide
1-[2-(2-aminoethyl)quinazolin-4-yl]-N,N-dipropylpiperidin-4-amine
2-(2-chloro-4-{[3-(dimethylamino)piperidin-1-yl]methyl}-6-methoxyphenoxy)acetamide
methyl (2S)-2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}-3-methylbutanoate
1-ethyl-4-({2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-indole
4-[(dimethylamino)methyl]-4-hydroxy-N-[2-(1H-pyrazol-1-yl)phenyl]azepane-1-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-(3-chlorophenyl)-N-methyl-1,2,4-triazin-3-amine
1-methyl-4-{1-[5-(6-methylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]butan-2-yl}piperazine
4-(4-chlorophenoxy)-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine
5-ethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)thiophene-3-sulfonamide
4-[4-(2-methoxyphenyl)piperidin-1-yl]-2-(trifluoromethyl)pyrimidine
3-[(4S)-2,5-dioxoimidazolidin-4-yl]-N-[1-(4-fluorophenyl)piperidin-4-yl]propanamide
N,N-dimethyl-5-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
(2S,4S)-4-(benzylamino)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-methoxy-5-{[8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
(1H-1,3-benzodiazol-2-ylmethyl)(2-methoxyethyl)[(4-methylphenyl)methyl]amine
N-benzyl-3-{[3-(methoxymethyl)piperidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)pyrimidin-5-yl]acetic acid
5-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N2-benzyl-6-(3,5-difluorophenyl)-1,3,5-triazine-2,4-diamine
1-({3-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
6-methyl-N4-[3-(morpholin-4-yl)propyl]pyrimidine-2,4-diamine
6-[(2-methoxypyridin-3-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
(1S,5S)-N-[6-(3-methoxyphenoxy)pyridin-3-yl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(1R,3S)-7-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
N-(1-cycloheptylpiperidin-3-yl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-3-carboxamide