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4-[3-(1-ethyl-1H-pyrazol-4-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]benzoic acid
2-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
(2E)-1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)prop-2-en-1-one
methyl 4-(4-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
5-methoxy-3-methyl-2-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1H-indole
9-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}but-2-yn-1-one
4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-(2-methoxyethyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
4-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
2-(4-ethylpiperazin-1-yl)-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]ethan-1-one
(1R,9S)-5-amino-3-[2-(2-methylphenyl)pyrimidin-5-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
1-(2-methoxyethyl)-3-(2-methylpropyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[5-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)furan-2-yl]-1H-pyrazole
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(pyridin-3-yl)piperazine
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-(4-phenoxybenzoyl)piperidine
3-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]phenyl}-N-methylpropanamide
N-[(4-hydroxyphenyl)methyl]-2,6-dimethyl-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide
1-[(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2-[4-(4-butylpiperazine-1-carbonyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
4-(hydroxymethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
N-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-methyl-5-{1-[2-(thiophen-2-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(3-chloropyridin-2-yl)piperidin-4-yl]propanamide
6-tert-butyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(butan-2-yl)-5-chloro-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
5-ethyl-2-methyl-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
(4aS,8aR)-1-(2-aminoethyl)-6-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
methyl 4-{[(2-{5-oxo-1-[(1-phenylcyclopentyl)methyl]pyrrolidin-2-yl}ethyl)amino]methyl}benzoate
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[3-(oxolan-2-yl)propyl]amine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
2-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-ol
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-methoxyethan-1-one
4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
4-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-fluoropyridine
5-[4-(benzenesulfonyl)phenyl]-1,2,3,4-tetrahydroisoquinoline
N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]-3-(2-oxopiperidin-1-yl)propanamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-methoxypropan-1-one
(1S,5R)-3-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-N,8-dimethyl-2-[2-(pyridin-4-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-benzyl-9-[(2S)-3-hydroxy-2-methylpropyl]-2,9-diazaspiro[5.5]undecan-3-one
N-phenyl-5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazole
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-phenyl-1,2,3,6-tetrahydropyridine
N-(1-methyl-1H-pyrazol-5-yl)-3-({methyl[(3-methyloxetan-3-yl)methyl]amino}methyl)benzamide
2-amino-6-(4-ethylphenyl)-4-(2-methyl-1H-imidazol-4-yl)pyridine-3-carbonitrile
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
2-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
2-(3-methoxypiperidin-1-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
1-[(4aR,8aR)-4a-hydroxy-7-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]ethan-1-one