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1-[(4-methylphenyl)methyl]-5-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}pyrrolidine-3-carboxamide
N-[3-(6-phenylpyridazin-3-yl)phenyl]acetamide
2-methyl-4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}-1,2-dihydrophthalazin-1-one
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-(quinolin-3-yl)urea
[(4-ethylphenyl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-ethyl-4-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1H-indole
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(pyrazin-2-yl)propanamide
2-(1-benzofuran-2-yl)-3-(piperidine-1-carbonyl)pyridine
3-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(propan-2-yl)piperazine-1-carboxamide
(3S,4R)-3-benzyl-4-methyl-1-(quinoline-3-carbonyl)piperidin-4-ol
1-(carbamoylmethyl)-N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-4-carboxamide
N-[1-(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)pyrrolidin-3-yl]acetamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(methoxymethyl)furan-2-carboxamide
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(2-methylpropyl)piperidine
N-cyclobutyl-3-{[1-(1H-pyrazol-1-yl)propan-2-yl]sulfamoyl}benzamide
[(1-cyclopentylpiperidin-3-yl)methyl][2-(piperidin-1-yl)ethyl](1,3-thiazol-4-ylmethyl)amine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(3,3,3-trifluoropropyl)-1,4-diazepan-5-one
3-(2H-1,3-benzodioxol-5-yl)-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(2R)-2-(hydroxymethyl)-N-[2-methoxy-5-(methylcarbamoyl)phenyl]pyrrolidine-1-carboxamide
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(propyl)amino]methyl}phenoxy)propan-2-ol
(2R,3R,6R)-5-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1r,4r)-4-hydroxycyclohexyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-{4-[1-(2-methylfuran-3-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
2-benzyl-9-(3-propyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(1,4-dimethylpiperazin-2-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
5-methyl-N4-{2-[methyl(phenyl)amino]ethyl}pyrimidine-2,4-diamine
3-methyl-N-[(5-methylpyrazin-2-yl)methyl]-5-(phenoxymethyl)furan-2-carboxamide
methyl (2S)-2-[(1-cyclohexyl-1H-1,2,3-triazol-4-yl)formamido]-3-(1H-imidazol-4-yl)propanoate
2-(3-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(2-phenylethyl)-3,4-dihydropyrimidin-4-one
N-(4-{2-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]acetamido}phenyl)-N-methylacetamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole
4-benzyl-3-(1-cyclopentylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4-ethylphenyl)methyl]-3-(2-hydroxypyridin-3-yl)-1-(2-methoxyethyl)urea
(1S,5R)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
2-[(5-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
{[6-(3-chloro-5-fluorophenyl)pyridin-3-yl]methyl}dimethylamine
(5S,9aS,9bS)-5-(2-fluorophenyl)-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(2-methoxyethyl)-2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(propan-2-yl)acetamide
1-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)imidazolidin-2-one
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
2-phenoxy-N-{4-[4-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]phenyl}acetamide
4-(1-methylcyclopropanecarbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-ethoxy-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]acetamide
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(methylsulfanyl)ethan-1-one
7-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[3-({2-[(4-fluorophenyl)methyl]morpholin-4-yl}methyl)phenyl]ethan-1-one
N-[2-(oxan-3-yl)ethyl]-6-(piperidin-1-yl)pyrimidin-4-amine
2-chloro-N-(2-{[2-(methylamino)pyrimidin-5-yl]formamido}ethyl)benzamide
1-{4-[(2-ethylpyrimidin-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2,2-dimethylpropan-1-one