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1-(1-ethylpiperidin-4-yl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
5-[2-(oxan-2-ylmethoxy)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
6-{4-[(6-ethoxypyridin-3-yl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)furan-2-carboxamide
2-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-cyclohexyl-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-ethyl-1H-pyrazole
2-{4-[3-(morpholine-4-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenol
2-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-6-methoxyphenol
4-{2-[(2-methoxyphenyl)methoxy]phenyl}-1,5-dimethyl-1H-pyrazole
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-phenylbenzoyl)piperidine
(2R)-2-amino-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(1H-indol-3-yl)propan-1-one
5-methyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-3-[3-(2,4-difluorophenyl)propanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]hexanoic acid
2-[2-({[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]urea
6-[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
3-(4-chloro-2-methylbenzoyl)piperidine
3-(2-ethoxyphenyl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
2-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[3-(morpholin-4-yl)propyl]pyrrolidin-2-one
6,7-dimethyl-2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-1,3-benzodiazole
2-{[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
3-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-N,N-dimethylpropanamide
N-[(3S,4R)-1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-[5-cyclopropyl-4-(2-methylpiperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(2-methoxyphenyl)pyrimidine
2-{5-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
6-({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)pyridine-3-carbonitrile
N-[(1-cycloheptylpyrrolidin-3-yl)methyl]-2-methoxybenzamide
2-(1-{1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
2-[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-4-carbonitrile
2-[cyclohexyl(methyl)amino]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}propanamide
(3S,4R)-4-(3-fluorophenyl)-1-(3,3,3-trifluoropropyl)pyrrolidine-3-carboxylic acid
N-[3-(4H-1,2,4-triazol-4-yl)phenyl]azocane-1-carboxamide
2-chloro-5-[({2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}carbamoyl)amino]-N,N-dimethylbenzamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-(quinolin-6-ylmethyl)piperidine-3-carboxamide
4-methyl-4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}piperidine
1-methyl-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-cyclopropanecarbonyl-3-[2-(2-methylphenyl)ethyl]piperidine
6-fluoro-2-methyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)quinoline-4-carboxamide
9-(oxolan-3-ylmethyl)-2-[2-(1H-pyrazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-[4-(quinolin-3-yl)phenyl]acetamide
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[2-(phenylsulfanyl)ethyl]piperidine
[(1-butyl-1H-1,2,4-triazol-5-yl)methyl](methyl)(pyridin-2-ylmethyl)amine
3-(methylsulfanyl)-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]propanamide
[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl][1-(methylsulfanyl)propan-2-yl]amine