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1-(1-{5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperidin-4-yl)piperidin-3-ol
(benzylsulfamoyl)({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
(2S,4S)-4-amino-N-methyl-1-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]pyrrolidine-2-carboxamide
5-(4-fluorophenyl)-N-(2-methanesulfonylethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
1-(propan-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(dimethylamino)ethyl]methylamine
2-[(3,5-dimethoxyphenyl)methyl]-2-azaspiro[4.4]nonan-3-one
3-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methoxypyridine
N-{2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}-1H-pyrrole-2-carboxamide
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
1-{4-[(2-propoxyethyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
4-phenyl-3-[1-(2-phenylethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-ethyl-N-[3-(furan-2-amido)-4-methoxyphenyl]-3-methylpiperidine-3-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-{[4-(thiophene-2-carbonyl)piperazin-1-yl]methyl}quinazolin-4-amine
3-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-chloro-1,2-dihydropyridin-2-one
N5-cyclopropyl-N6-[(2-methyl-1,3-thiazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-{2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
3-methyl-N-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
3-({[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)-4H-chromen-4-one
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-4-methoxyphenol
2-methoxy-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3-{2-[1-(2-ethylpyridine-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(2-fluorophenyl)-5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
2-(morpholin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-methoxy-N-[2-methyl-3-({[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]carbamoyl}amino)phenyl]acetamide
3-methyl-1-{1-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
N-{3-[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-3-oxopropyl}methanesulfonamide
N-[(2-chloropyridin-3-yl)methyl]-N,5-dimethyl-2-(2-methylpropanamido)benzamide
3-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-1,2,3,4-tetrahydroisoquinoline
(4aS,7aR)-1-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,5R)-1-[2-(3-chloro-4-hydroxyphenyl)acetyl]-5-(cyclopropylcarbamoyl)piperidine-3-carboxylic acid
5-({methyl[(3-{2-[4-(3-phenyl-1,2-oxazole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
3-(azocan-1-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)propanamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-(methylsulfanyl)pyrimidin-4-amine
4-(3-benzyl-1H-1,2,4-triazol-5-yl)-2,6-dimethoxypyrimidine
6-cyclopentyl-N-[2-(ethylsulfanyl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-{2-oxa-7-azaspiro[4.5]decane-7-sulfonyl}-1,2,3,4-tetrahydroquinolin-2-one
1-[9-hydroxy-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
2-{1-[1-(2,3,6-trifluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
1-[(3-chlorophenyl)methyl]-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
(3S)-2-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylic acid
N-(2-{1-[3-(1-hydroxyethyl)phenyl]-1H-imidazol-4-yl}ethyl)acetamide
4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-{1-[1-(3-hydroxypropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
3-{[cyclohexyl(methyl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
(2R,6S)-2,6-dimethyl-4-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)morpholine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide