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N-benzyl-3-cyclopropyl-N-(3-hydroxy-2-methylpropyl)propanamide
N-[2-(benzyloxy)ethyl]-5-tert-butyl-1,3,4-oxadiazol-2-amine
2-amino-4-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-6-(pyridin-3-yl)pyridine-3-carbonitrile
{3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-2,2-dimethylpropyl}dimethylamine
4-[(2-amino-5-ethylpyrimidin-4-yl)amino]-1-(4-fluorophenyl)pyrrolidin-2-one
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[(4-methylphenyl)sulfanyl]piperidine
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethylbenzamide
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidine
(2S,4S)-N-ethyl-1-(pyridin-2-ylmethyl)-4-[(quinoxalin-2-yl)amino]pyrrolidine-2-carboxamide
2-[(4-chlorophenyl)methyl]-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
6-cyclopentyl-N-(2-hydroxy-3-methoxypropyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-(3-chlorophenyl)-9-methoxy-4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
4-{1-[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-oxopropan-2-yl}-1,2-dihydrophthalazin-1-one
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
5-methyl-N4-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidine-2,4-diamine
N-[(3S,4R)-1-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-methyl-2-{4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}acetamide
1-[3-(2-fluorophenoxy)azetidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
3-(2-aminoethyl)-4-(4-chlorophenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,7S,8aS)-7-{[(2-fluorophenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-[(4-phenylphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-oxo-1-(2-phenylethyl)-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
(1R,5R)-3-(5-chlorothiophene-2-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
5,7-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyrido[2,3-d]pyrimidin-4-amine
[(2-chlorophenyl)methyl]({[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
4-(3-methoxyphenyl)-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]benzamide
1-(2,3-dimethylquinoxalin-6-yl)-3-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]urea
1,3-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-({2-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)piperazin-1-yl]ethan-1-one
(1S,5R)-3-[2-(3-fluorophenyl)ethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-amino-4-(3,4-dihydroxyphenyl)-6-(3-methylphenyl)pyridine-3-carbonitrile
2-(1H-imidazol-1-yl)-1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]ethan-1-one
2-{[4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
N-ethyl-4-methyl-5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
3-{3-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propyl}pyridine
1-[(5-ethylfuran-2-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-4-(6-methoxypyridin-2-yl)phenol
benzyl N-[1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)pyrrolidin-3-yl]carbamate
N-[2-(2-chlorophenyl)-1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-[2-(pyrrolidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
8-(2-butoxyacetyl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(1,4-diazepane-1-carbonyl)-N-(pyridin-3-ylmethyl)benzene-1-sulfonamide
{5-[3-(5-methylfuran-2-yl)-1-propyl-1H-1,2,4-triazol-5-yl]-1H-1,3-benzodiazol-2-yl}methanol
4-[1-(pyridin-3-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one