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1-ethyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-6-oxopiperidine-3-carboxamide
1-{6-hydroxy-4-[2-(methylsulfanyl)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
4-(pyridin-3-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}pyrimidin-2-amine
3-methoxy-1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)pyrrolidine
5-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
2-(ethoxymethyl)-N-(prop-2-en-1-yl)-7-(pyridin-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(2,4-dioxoimidazolidin-1-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-fluorophenoxy)ethan-1-one
3-(azocan-1-yl)-N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]propanamide
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{5-[(4-acetamidopiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
3-({[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
N-cyclopentyl-1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
(4S)-1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
5-chloro-N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-3-methyl-N-(oxolan-2-ylmethyl)-1H-indole-2-carboxamide
1-(2-methylphenyl)-4-[4-(piperidin-1-ylmethyl)benzoyl]-1,4-diazepane
{[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]sulfamoyl}(ethyl)methylamine
5-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-2-methylpyrimidine
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
3-ethyl-4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1-methylpiperazin-2-one
2-[2-(1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
2-{2-[(thiolan-3-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
1-[2-(3-fluorophenyl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
4-(2-cyclopropyl-1H-imidazol-1-yl)-2,3-dimethylphenol
methyl (2S)-3-methyl-2-({1-[4-(2-phenoxyacetamido)phenyl]piperidin-4-yl}amino)butanoate
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
7-(1,3-benzothiazol-2-yl)-4-[(2-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(6-methoxynaphthalen-2-yl)-4-(2-methoxypyridine-4-carbonyl)morpholine
2-(2-fluorophenyl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{[5-(3-chloro-4-methylphenyl)furan-2-yl]methyl}-4-methoxypiperidine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
4-cyano-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-4-phenylpiperidine-1-carboxamide
2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-N-(5-methyl-1,2-oxazol-3-yl)-2-oxoacetamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-(pyridin-2-ylsulfanyl)acetamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-phenylbenzamide
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2-methyl-3,4-dihydropyrimidin-4-one
(butan-2-yl)[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](pyridin-4-ylmethyl)amine
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-(2-methylphenyl)propan-1-one
3-(1-benzylpiperidin-3-yl)-1-[2-(dimethylamino)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-cyclopentyl-5-(2-methyl-6-propylpyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-9-(1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-({[1-(9H-purin-6-yl)piperidin-4-yl]amino}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-{[(3-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3S,4R)-1-(2-ethoxypyridine-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-(1-methylpiperidin-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
1-({1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
4-(4-methoxypyrimidin-2-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol