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5-{[benzyl(methyl)amino]methyl}-N-[1-(pyridin-4-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-[(2-fluorophenyl)methyl]-1-[2-(piperidin-1-yl)ethyl]piperidine
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
8-(oxan-3-yl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-phenyl-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2,3,6-tetrahydropyridine
2-(furan-2-yl)-5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
2-{3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-1H-imidazole
N-[(3R,4S)-1-(2-aminopyridine-4-carbonyl)-4-cyclopropylpyrrolidin-3-yl]methanesulfonamide
3-(2,4-dichlorophenyl)pyridin-4-amine
2-(2-methoxyethyl)-4-(piperidin-4-ylmethyl)morpholine
(2R)-2-amino-N,4-dimethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pentanamide
(2R)-2-{5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}propanamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]acetamide
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(pyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-methoxyquinazolin-6-yl)aniline
(1S,5R)-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-methylpiperidine
5-methyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
2-(3-acetyl-7-ethyl-1H-indol-1-yl)-1-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl][(2-fluoro-5-methoxyphenyl)methyl]methylamine
2-cyclopropyl-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-[(3,4-difluorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methylpiperidine-2-carboxamide
5-[(3-chloro-2,6-difluorophenyl)methyl]-3-methyl-1-propyl-1H-1,2,4-triazole
1-(2-fluorophenyl)-2-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-[3-(1H-imidazol-1-yl)propyl]-9-(6-methylpyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[(4-benzylpiperidin-1-yl)methyl]-N-ethyl-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-1-methyl-1H-1,3-benzodiazole
2-(4-methyl-1H-imidazol-5-yl)-1-[2-(5-methylfuran-2-yl)ethyl]-1H-imidazole
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-2-carboxamide
3-(pyridin-2-yl)-N-[1-(thiophen-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
5-tert-butyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3,4-oxadiazol-2-amine
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-methyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-2-(thiophen-2-ylformamido)propanamide
2-(4-methyl-1H-imidazol-5-yl)-1-{1-oxaspiro[4.4]nonan-3-yl}-1H-imidazole
2-(3-methoxypropyl)-9-(quinoxaline-6-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-10-oxo-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-[3-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
N-(4-methoxyphenyl)-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-3-amine
2-{3-[(cyclobutylamino)methyl]-2-methyl-1H-indol-1-yl}acetamide
2-(1-benzylpiperidin-4-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
1-(4-ethylpiperazin-1-yl)-3-{1-[(2R)-2-hydroxy-2-phenylacetyl]piperidin-4-yl}propan-1-one
(4aS,8aR)-6-(1H-1,3-benzodiazole-5-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
4-hydroxy-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
6-[(5-acetamidothiophen-2-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[3,5-dimethyl-4-(5-methyl-1H-indol-3-yl)-1H-pyrazol-1-yl]propanamide