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4-methyl-2-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
7-(3,6-dimethylpyrazin-2-yl)-4-[3-(methylsulfanyl)butyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
5-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
(2R,6R)-4-cycloheptanecarbonyl-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[2-(benzenesulfonyl)ethyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-(pyridin-3-ylmethyl)-4-(4,5,6-trimethylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 4-{[4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzoate
6-{[(cyclopentylmethyl)(methyl)amino]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methylbut-2-en-1-one
1-[(2-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-pyrazole
1-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-yl)piperidin-3-ol
2,6-dimethyl-3-(morpholine-4-carbonyl)quinoline
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2,2,2-trifluoroethyl)acetamide
4-[5-(1H-indol-2-yl)-4-phenyl-1H-imidazol-1-yl]-N,N-dimethylbutanamide
1-(2-propyl-1,3-thiazole-4-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-6-methoxypyrimidin-4-amine
1-[3-(azetidine-1-sulfonyl)benzoyl]-3-(methoxymethyl)pyrrolidine
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(4-{4-[(3,3-diphenylpropyl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-(thiophene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
ethyl 1-(1,4-dithiepan-6-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-4-(4-fluorophenyl)-1,3-thiazole
(4aS,8aR)-6-[(2-methylphenyl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
N-(2-chloropyridin-3-yl)-4-(furan-2-carbonyl)-1,4-diazepane-1-carboxamide
2-[3-(2-methoxypyridin-3-yl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-[(6-methylpyridin-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
4-[3-(1H-pyrazol-1-ylmethyl)benzamido]oxane-4-carboxylic acid
3-(4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazin-1-yl)-1,2-benzothiazole
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-6-sulfonamide
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]benzamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(morpholin-3-yl)ethan-1-one
N-[3-(4-oxo-4H-chromen-3-yl)phenyl]acetamide
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-3,4-dihydroquinazolin-4-one
9-{2-[methyl(propan-2-yl)amino]acetyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
4-[1-(1,3-thiazol-4-ylmethyl)piperidin-4-yl]pyrimidine
8-[(1-cyclopropylethyl)amino]-2,6-dimethyloctan-2-ol
6-(4,4-dimethylpiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(4aS,8aS)-2-[2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-decahydroisoquinolin-4a-ol
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
1-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
4-(1H-indazole-3-carbonyl)-1-(2-methylphenyl)piperazin-2-one
2-oxo-1-(2-phenylethyl)-3-(pyrimidin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
4-(2-methyl-1,3-thiazole-4-carbonyl)-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine