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4-(2,6-dimethylpyridin-3-yl)-6-methoxypyrimidin-2-amine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-methyl-9-[3-(pyridin-3-yl)propanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-[(1S,5R)-6-[(5-acetylthiophen-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}propanamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(oxan-4-yl)piperidine
6-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-(2-phenylethyl)piperidine-3-carboxamide
(4aS,7aR)-1-(4-methyl-1H-pyrrole-2-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(4-chlorophenyl)sulfanyl]-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]pyrazine
N-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazole-5-carboxamide
{4-[(4-pentyl-1H-1,2,3-triazol-1-yl)methyl]phenyl}methanol
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
5-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
6-methyl-4-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[2-(1H-imidazol-4-yl)ethyl]-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
1-(2,3-dihydro-1H-inden-5-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-cyclopropyl-5-(3-acetamidophenyl)furan-2-carboxamide
[2-(3,4-dimethylphenoxy)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-[(4-chlorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]piperidin-3-amine
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
(4aR,7aS)-1-ethyl-4-[4-(1,3-oxazol-5-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(3-chlorophenyl)-4-(2-methylpyrimidine-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[2-(azepan-1-ylmethyl)phenyl]-6-(4-fluorophenyl)-3,4-dihydropyrimidin-4-one
8-(3-ethoxybenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(1-benzofuran-2-ylmethyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-3-[(5-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}furan-2-yl)sulfanyl]-4H-1,2,4-triazole
(2R,6R)-4-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
3-{[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}benzoic acid
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl][3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]methylamine
1-[(4-methoxyphenyl)methyl]-4-[3-(pyridin-3-yl)propanoyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-ethyl-4-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}pyrimidine
(2R,3R)-3-amino-1'-[6-(trifluoromethyl)pyridin-2-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1,2-dihydroquinazolin-2-one
N5-[(4-chlorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-fluoro-N-(2-hydroxyethyl)-6-methoxy-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
1-methyl-3-(2-methylpropyl)-N-(1,2-oxazol-5-ylmethyl)-1H-pyrazole-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[5-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]azetidine-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-N'-phenylethanediamide
4-{[1-(5-phenoxyfuran-2-carbonyl)piperidin-4-yl]methyl}morpholine
5-(1-ethyl-1H-imidazol-5-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
methyl (1R,3S,3aR,6aS)-5-methyl-4,6-dioxo-1-(propan-2-yl)-3-(quinoxalin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-[1-(1-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]benzoic acid
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7,7-dimethyl-2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one