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2-{3-[(2,2-dimethylmorpholin-4-yl)methyl]phenyl}-6-phenyl-3,4-dihydropyrimidin-4-one
N-[(2-{4-[3-(4-methoxyphenyl)propanamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1-methylpiperidine-2-carboxamide
2-methyl-5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-methyl-N-[2-(oxan-2-yl)ethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
methyl (2S)-2-{[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}-4-methylpentanoate
8-(2,2,3-trimethylbut-3-enoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(2-methoxybenzamido)phenyl]-6-oxopiperazine-2-carboxamide
N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(2S)-1-(dimethyl-1,3-thiazole-5-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
4-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
N-benzyl-1-(propan-2-yl)-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1H-indazole
6-(dimethylamino)-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}pyridine-3-carboxamide
N-methyl-3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-[(4-fluorophenyl)methyl]-N,2-dimethyl-1-benzofuran-7-carboxamide
4-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(3aR,6aR)-2-acetyl-5-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclopropanecarbonyl-8-(3,4-dimethylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(1-ethylpiperidin-4-yl)-N-[1-(4-fluorophenyl)propyl]acetamide
1-ethyl-8-[(4-hydroxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
3-[2-(dimethylamino)ethyl]-5-[1-(3-methoxybenzoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-imidazol-1-yl)propan-1-one
1-ethyl-5-(4-methylpiperidin-1-yl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-fluoro-N-(1H-indol-5-ylmethyl)-5-sulfamoylbenzamide
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-ethylpiperazine
1-ethyl-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
[1-(5-chloro-2-fluorobenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-3-amine
5-hydroxy-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrazine-2-carboxamide
1-cyclohexyl-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-1,7-dimethyl-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
4-{[2-(3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
methyl 3-[1-(2-hydroxy-2-phenylethyl)-1H-imidazol-2-yl]benzoate
3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]-1-(1,4-oxazepan-4-yl)propan-1-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-(3-chloro-4-methoxybenzoyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
5-ethyl-4-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}pyrimidin-2-amine
(3R,4R)-3-methyl-1-(3-methylpyrazin-2-yl)-4-(oxan-4-yl)piperidin-4-ol
1-[(2,3-dichloro-4-methylphenyl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
methyl 4-(5-methyl-4-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-1,3-oxazol-2-yl)benzoate
1-(2-chlorophenyl)-4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperazin-2-one
1-({5-[2-(3-fluorophenyl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
6-(azepan-1-yl)-N-methyl-N-(oxolan-3-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidin-3-yl]methanol