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1-{1-[(5-butylthiophen-2-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,1-dioxo-1λ6-thiane-4-carboxamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methylacetamide
4-{[2-(5-chloro-1,2,4-thiadiazol-3-yl)phenyl]methyl}morpholine
methyl 1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-phenylpyrrolidine-3-carboxylate
5-(propan-2-yl)-N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-chloro-N-[2-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-({4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-4-methoxyphenol
8-(1-methyl-1H-pyrazole-3-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-methoxyethyl)-9-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-butyl-2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
2-(5-methyl-1H-pyrazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
5-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
5-[benzyl(methyl)amino]-2-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-2,3-dihydropyridazin-3-one
(1S,5R)-3-[(4-chlorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N,2-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-{3-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
1-{6-[4-(2-phenoxyethyl)piperazin-1-yl]pyridin-2-yl}ethan-1-ol
N-[(4-fluorophenyl)methyl]-3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]propanamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
3-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-1H-indazole
1-(2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(2-methylphenyl)methyl]piperazine
N3-[2-(5-methoxy-1H-indol-3-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-{1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
4-(1-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-1H-imidazol-2-yl)benzoic acid
8-(5-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
8-(5-cyano-2-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-4,6-dimethylpyridine-3-carbonitrile
2-[2-(2-phenylethyl)morpholine-4-carbonyl]-1,4-dihydroquinolin-4-one
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(furan-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N,N-dimethyl-2-[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]propanamide
1-(2-methoxyphenyl)-4-(1-methylpiperidine-2-carbonyl)piperazin-2-one
(4aS,7aR)-N-(3-ethylphenyl)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-[5-(2,3-dimethylphenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(1-benzothiophene-5-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
(1S,5R)-6-methyl-3-(2-phenylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-4-(4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}phenyl)butan-2-ol
1-(pyridin-2-yl)-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(1-methylpyrrolidin-2-yl)acetamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dimethylacetamide
1-[4-(3-chlorophenyl)piperazin-1-yl]-2-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)-4-phenylphenoxy]ethan-1-one
3-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}-N-(2-methylphenyl)propanamide
ethyl 2-(1H-indol-5-yl)pyridine-3-carboxylate
2-methyl-3-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1H-indole-5-carbonitrile