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3-chloro-4-({1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
1-(diphenylmethyl)-4-(4-methyl-1H-imidazole-5-carbonyl)piperazine
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[2-methyl-2-(pyrrolidin-1-yl)propyl]acetamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
4-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-4-oxobutanamide
3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2,5-dimethylpyrazine
4-{[methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
N-cyclopentyl-2-(furan-2-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxoacetamide
3-(3-chlorophenyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-3-phenylpropanamide
2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propane-1,3-diol
5-(2-hydroxy-4-methylpentanoyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-(2-{2-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)acetamide
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
(4aS,8aR)-1-(3-hydroxypropyl)-6-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
2-{4-[2-(3-methyl-2-oxopyrrolidin-1-yl)acetyl]piperazin-1-yl}benzonitrile
N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
2-fluoro-N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]benzamide
ethyl 3-[(4-fluorophenyl)methyl]-1-(isoquinoline-3-carbonyl)piperidine-3-carboxylate
3-(2H-1,3-benzodioxol-5-yl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-phenylpropanamide
8-methyl-2-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]-2,8-diazaspiro[4.5]decan-3-one
N-{4-[({2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}carbamoyl)methoxy]phenyl}propanamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-amine
3-propyl-5-[4-(1,2,3-thiadiazol-4-yl)phenoxymethyl]-1,2,4-oxadiazole
3-[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl]-4-[(2-ethoxyphenyl)methyl]piperazin-2-one
4-({5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
1-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
methyl 4-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]carbamoyl}butanoate
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{2-[(2-chlorophenyl)formamido]ethyl}-4-(1H-pyrazol-4-yl)butanamide
1-{1-[5-(methoxymethyl)furan-2-carbonyl]azetidin-3-yl}-2-methylpiperidine
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
3-(2-methoxyethyl)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidine-3-carboxylic acid
N-[1-(2-methoxyethyl)-7-(4-phenylpiperazine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
5-(oxolan-3-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
N-[(5-{[3-(butan-2-yloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
6-{[5-(1-ethylpiperidin-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyrimidin-4-ol
N-methyl-3-(5-methylfuran-2-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-(3,4-difluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
2-(morpholin-2-yl)-N-(3-phenylprop-2-yn-1-yl)-N-propylacetamide
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
N-cyclopropyl-1-[1-(4-methylquinolin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
2-(5-methoxypyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-[methyl(phenyl)amino]ethan-1-one
2-amino-6-hydroxy-4-[2-(2-hydroxyethoxy)phenyl]-5H-indeno[1,2-b]pyridine-3-carbonitrile
2-(2-phenylethyl)-1-(pyrrolidine-1-sulfonyl)piperidine