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N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylbutanamide
5-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-(2-ethoxyethyl)-3-methyl-1H-pyrazole
1-(cyclohex-3-ene-1-carbonyl)-4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
N-(3-chloro-4-propoxyphenyl)-3-(pyridin-3-yl)azetidine-1-carboxamide
N-[2-ethyl-4-(2-propyl-1H-imidazol-1-yl)phenyl]acetamide
6-(3-fluoro-4-methoxyphenyl)-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-1-(pyrimidin-2-yl)piperidin-4-amine
3-({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)-N-(pyridin-3-yl)propanamide
N-benzyl-N-methyl-3-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}propanamide
3-[(3-phenylprop-2-yn-1-yl)(propyl)amino]propane-1,2-diol
1-methyl-4-phenyl-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-methylpyridin-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine
8-[5-(propan-2-yl)pyrimidin-4-yl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-8-[4-(1H-pyrazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-{[3-(1H-pyrazol-4-yl)phenyl]formamido}ethyl)acetamide
2-(2-ethyl-1H-imidazol-1-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
3-({1-[2-(methylamino)acetyl]pyrrolidin-3-yl}methyl)benzamide
N-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-2,6,8-trimethylquinoline-4-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
8-methoxy-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[5-chloro-2-(propan-2-yloxy)phenyl]methyl}-2-(1H-imidazol-2-yl)benzamide
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-3-(pyrazin-2-yl)propan-1-one
2-(3-hydroxyphenyl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-cyclohexyl-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
1-{2-[1-(6-methyl-1,3-benzothiazol-2-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
(1S,5R)-3-(2-ethylpyridine-4-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-chloro-N-[3-(1H-indol-1-yl)propyl]-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-5-[2-(2-{[5-(propan-2-yl)pyrimidin-4-yl]amino}ethyl)morpholin-4-yl]-2,3-dihydropyridazin-3-one
2-methyl-3-(2-oxo-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(2R)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenylbutan-1-one
1-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4-[2-(propan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
[(2-ethylpyrimidin-5-yl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
1-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(thian-4-yl)piperazine
2-{4-[1-(dimethylamino)ethyl]phenyl}-5,6-dimethylpyridine-3-carbonitrile
N-{3-[3-(1-phenylcyclobutyl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
2-{1-[2-(hydroxymethyl)phenyl]-1H-pyrazol-4-yl}ethan-1-ol
{1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
1-(2-methoxyethyl)-4-[3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]pyrrolidin-2-one
1-[cyclohexyl(methyl)amino]-3-[3-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
6-(3-hydroxyazetidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}-N,N-bis(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(2,5-difluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide