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8-(1-ethyl-1H-pyrazole-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(2-methylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
1-{1-[3-(4-hydroxyphenyl)benzoyl]piperidin-4-yl}piperidin-4-ol
4-{[1-(1,1-dioxo-1λ6-thiane-4-carbonyl)piperidin-3-yl]methyl}benzoic acid
{[4-(4,6-dimethoxypyrimidin-2-yl)phenyl]methyl}dimethylamine
(2S)-2-acetamido-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)propanamide
3-chloro-4-fluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-N-(trimethyl-1H-pyrazol-4-yl)benzamide
N,N-dimethyl-2-(4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)acetamide
2-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}-2-(4-fluoro-3-methylphenyl)acetic acid
N-cyclopropyl-8-methoxy-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-[(diethylamino)methyl]-N-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1,4-diazepane
5-{[(2-fluorophenyl)methyl]amino}-1-methyl-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-benzyl-5-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
1-(carbamoylmethyl)-N-[1-(6-methoxynaphthalen-2-yl)ethyl]piperidine-4-carboxamide
N-(2,4-dimethoxyphenyl)-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propanamide
2-methyl-6-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
2-(2-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)-4-methoxy-6-methylpyrimidine
2-oxo-8-{[(2-phenylethyl)carbamoyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-cyclopropyl-1-[(1s,4s)-4-[2-(2-chlorophenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3S)-3-(dimethylamino)azepan-1-yl]propan-1-one
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-(4-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}thiophen-2-yl)ethan-1-one
N-[1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
N-benzyl-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
(3-cyclopentylpropyl)[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
{3-[(2-methylphenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-yl}methanol
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-methoxy-2-methylpropanamide
(1R,2R,6S,7S)-4-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
2-{4-[(3,5-dichloropyridin-4-yl)methyl]piperazin-1-yl}pyrazine
4-{4-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperazin-1-yl}-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-(quinolin-6-ylmethyl)propanamide
2-[1-(3-methylbutyl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
{1-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclobutyl}methanol
N2-[(1S,3aS,6aS)-octahydropentalen-1-yl]-N4-(propan-2-yl)pyrimidine-2,4-diamine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-6-methyl-2-phenylpyrimidin-4-amine
[3-(cyclopropylmethyl)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]methanol
(1S,5R)-6-propyl-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
3-fluoro-N-({7-[3-(2-oxopyrrolidin-1-yl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-amino-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-6-(propan-2-yl)pyrimidine-4-carboxamide
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
4-{[6-(2,3-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}thiomorpholine
1-(4-methyl-1H-imidazole-5-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
benzyl(cyclopropylmethyl){[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}amine
N,N-dimethyl-3-[4-({[3-(oxolan-3-yl)propyl]carbamoyl}amino)phenyl]propanamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide